                         SEQUENCE LISTING

<110>  BicycleRD Limited
 
<120>  BICYCLIC PEPTIDE LIGAND DRUG CONJUGATES

<130>  BIC-C-P2903PCT

<150>  GB2016331.7
<151>  2020-10-15

<160>  6     

<170>  PatentIn version 3.5

<210>  1
<211>  14
<212>  PRT
<213>  Artificial

<220>
<223>  Synthetic Peptide

<400>  1

Cys Tyr Asn Glu Phe Gly Cys Glu Asp Phe Tyr Asp Ile Cys 
1               5                   10                  


<210>  2
<211>  17
<212>  PRT
<213>  Artificial

<220>
<223>  Synthetic Peptide


<220>
<221>  Xaa
<222>  (1)..(1)
<223>  Xaa is B-Ala

<220>
<221>  Xaa
<222>  (2)..(2)
<223>  Xaa is Sar10

<220>
<221>  Xaa
<222>  (8)..(8)
<223>  Xaa is 1Nal

<220>
<221>  Xaa
<222>  (16)..(16)
<223>  Xaa is tBuGly

<400>  2

Xaa Xaa Ala Cys Ala Asn Glu Xaa Ala Cys Glu Asp Phe Tyr Asp Xaa 
1               5                   10                  15      


Cys 
    


<210>  3
<211>  12
<212>  PRT
<213>  Artificial

<220>
<223>  Synthetic Peptide

<400>  3

Cys Val Pro Cys Ala Asp Phe Pro Ile Trp Tyr Cys 
1               5                   10          


<210>  4
<211>  15
<212>  PRT
<213>  Artificial

<220>
<223>  Synthetic Peptide


<220>
<221>  Xaa
<222>  (1)..(1)
<223>  Xaa is B-Ala

<220>
<221>  Xaa
<222>  (2)..(2)
<223>  Xaa is Sar10

<400>  4

Xaa Xaa Ala Cys Val Pro Cys Ala Asp Phe Pro Ile Trp Tyr Cys 
1               5                   10                  15  


<210>  5
<211>  15
<212>  PRT
<213>  Artificial

<220>
<223>  Synthetic Peptide


<220>
<221>  Xaa
<222>  (3)..(3)
<223>  Xaa is 1Nal

<220>
<221>  Xaa
<222>  (7)..(7)
<223>  Xaa is HArg

<220>
<221>  Xaa
<222>  (13)..(13)
<223>  Xaa is HyP

<400>  5

Cys Pro Xaa Asp Cys Met Xaa Asp Trp Ser Thr Pro Xaa Trp Cys 
1               5                   10                  15  


<210>  6
<211>  17
<212>  PRT
<213>  Artificial

<220>
<223>  Synthetic Peptide


<220>
<221>  Xaa
<222>  (1)..(1)
<223>  Xaa is B-Ala

<220>
<221>  Xaa
<222>  (2)..(2)
<223>  Xaa is Sar10

<220>
<221>  Xaa
<222>  (5)..(5)
<223>  Xaa is 1Nal

<220>
<221>  Xaa
<222>  (9)..(9)
<223>  Xaa is HArg

<220>
<221>  Xaa
<222>  (15)..(15)
<223>  Xaa is HyP

<400>  6

Xaa Xaa Cys Pro Xaa Asp Cys Met Xaa Asp Trp Ser Thr Pro Xaa Trp 
1               5                   10                  15      


Cys 
    


