                         SEQUENCE LISTING

<110>  Max-Planck-Gesellschaft zur Frderung der Wissenschaften 
       e.V.
 
<120>  Selective TMPRSS2 inhibitors and medical use thereof

<130>  GAR-P04249WO

<160>  2     

<170>  PatentIn version 3.5

<210>  1
<211>  241
<212>  PRT
<213>  Homo sapiens


<220>
<221>  PDB-ID-6N4T
<222>  (1)..(241)
<223>  Matriptase

<400>  1

Val Val Gly Gly Thr Asp Ala Asp Glu Gly Glu Trp Pro Trp Gln Val 
1               5                   10                  15      


Ser Leu His Ala Leu Gly Gln Gly His Ile Cys Gly Ala Ser Leu Ile 
            20                  25                  30          


Ser Pro Asn Trp Leu Val Ser Ala Ala His Cys Tyr Ile Asp Asp Arg 
        35                  40                  45              


Gly Phe Arg Tyr Ser Asp Pro Thr Gln Trp Thr Ala Phe Leu Gly Leu 
    50                  55                  60                  


His Asp Gln Ser Gln Arg Ser Ala Pro Gly Val Gln Glu Arg Arg Leu 
65                  70                  75                  80  


Lys Arg Ile Ile Ser His Pro Phe Phe Asn Asp Phe Thr Phe Asp Tyr 
                85                  90                  95      


Asp Ile Ala Leu Leu Glu Leu Glu Lys Pro Ala Glu Tyr Ser Ser Met 
            100                 105                 110         


Val Arg Pro Ile Cys Leu Pro Asp Ala Ser His Val Phe Pro Ala Gly 
        115                 120                 125             


Lys Ala Ile Trp Val Thr Gly Trp Gly His Thr Gln Tyr Gly Gly Thr 
    130                 135                 140                 


Gly Ala Leu Ile Leu Gln Lys Gly Glu Ile Arg Val Ile Asn Gln Thr 
145                 150                 155                 160 


Thr Cys Glu Asn Leu Leu Pro Gln Gln Ile Thr Pro Arg Met Met Cys 
                165                 170                 175     


Val Gly Phe Leu Ser Gly Gly Val Asp Ser Cys Gln Gly Asp Ser Gly 
            180                 185                 190         


Gly Pro Leu Ser Ser Val Glu Ala Asp Gly Arg Ile Phe Gln Ala Gly 
        195                 200                 205             


Val Val Ser Trp Gly Asp Gly Cys Ala Gln Arg Asn Lys Pro Gly Val 
    210                 215                 220                 


Tyr Thr Arg Leu Pro Leu Phe Arg Asp Trp Ile Lys Glu Asn Thr Gly 
225                 230                 235                 240 


Val 
    


<210>  2
<211>  371
<212>  PRT
<213>  Homo sapiens


<220>
<221>  PDB-ID-1Z8G
<222>  (1)..(371)
<223>  Serine protease hepsin

<400>  2

Asp Gln Glu Pro Leu Tyr Pro Val Gln Val Ser Ser Ala Asp Ala Arg 
1               5                   10                  15      


Leu Met Val Phe Asp Lys Thr Glu Gly Thr Trp Arg Leu Leu Cys Ser 
            20                  25                  30          


Ser Arg Ser Asn Ala Arg Val Ala Gly Leu Ser Cys Glu Glu Met Gly 
        35                  40                  45              


Phe Leu Arg Ala Leu Thr His Ser Glu Leu Asp Val Arg Thr Ala Gly 
    50                  55                  60                  


Ala Ala Gly Thr Ser Gly Phe Phe Cys Val Asp Glu Gly Arg Leu Pro 
65                  70                  75                  80  


His Thr Gln Arg Leu Leu Glu Val Ile Ser Val Cys Asp Cys Pro Arg 
                85                  90                  95      


Gly Arg Phe Leu Ala Ala Ile Cys Gln Asp Cys Gly Arg Arg Lys Leu 
            100                 105                 110         


Pro Val Asp Arg Ile Val Gly Gly Arg Asp Thr Ser Leu Gly Arg Trp 
        115                 120                 125             


Pro Trp Gln Val Ser Leu Arg Tyr Asp Gly Ala His Leu Cys Gly Gly 
    130                 135                 140                 


Ser Leu Leu Ser Gly Asp Trp Val Leu Thr Ala Ala His Cys Phe Pro 
145                 150                 155                 160 


Glu Arg Asn Arg Val Leu Ser Arg Trp Arg Val Phe Ala Gly Ala Val 
                165                 170                 175     


Ala Gln Ala Ser Pro His Gly Leu Gln Leu Gly Val Gln Ala Val Val 
            180                 185                 190         


Tyr His Gly Gly Tyr Leu Pro Phe Arg Asp Pro Asn Ser Glu Glu Asn 
        195                 200                 205             


Ser Asn Asp Ile Ala Leu Val His Leu Ser Ser Pro Leu Pro Leu Thr 
    210                 215                 220                 


Glu Tyr Ile Gln Pro Val Cys Leu Pro Ala Ala Gly Gln Ala Leu Val 
225                 230                 235                 240 


Asp Gly Lys Ile Cys Thr Val Thr Gly Trp Gly Asn Thr Gln Tyr Tyr 
                245                 250                 255     


Gly Gln Gln Ala Gly Val Leu Gln Glu Ala Arg Val Pro Ile Ile Ser 
            260                 265                 270         


Asn Asp Val Cys Asn Gly Ala Asp Phe Tyr Gly Asn Gln Ile Lys Pro 
        275                 280                 285             


Lys Met Phe Cys Ala Gly Tyr Pro Glu Gly Gly Ile Asp Ala Cys Gln 
    290                 295                 300                 


Gly Asp Ser Gly Gly Pro Phe Val Cys Glu Asp Ser Ile Ser Arg Thr 
305                 310                 315                 320 


Pro Arg Trp Arg Leu Cys Gly Ile Val Ser Trp Gly Thr Gly Cys Ala 
                325                 330                 335     


Leu Ala Gln Lys Pro Gly Val Tyr Thr Lys Val Ser Asp Phe Arg Glu 
            340                 345                 350         


Trp Ile Phe Gln Ala Ile Lys Thr His Ser Glu Ala Ser Gly Met Val 
        355                 360                 365             


Thr Gln Leu 
    370     


