                               SEQUENCE LISTING

<110> INTARCIA THERAPEUTICS, INC.
 
<120> LONG ACTING PEPTIDE TYROSINE TYROSINE (PYY) ANALOGS AND METHODS 
      OF USE

<130> 717120: 102487-058WO

<140> PCT/US2021/027759
<141> 2021-04-16

<150> 63/076,459
<151> 2020-09-10

<150> 63/011,649
<151> 2020-04-17

<160> 814   

<170> PatentIn version 3.5

<210> 1
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 1
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Tyr 
        


<210> 2
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 2
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Tyr 
        


<210> 3
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 3
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Tyr 
        


<210> 4
<211> 35
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (35)..(35)
<223> n-methylY

<400> 4
Lys Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp 
1               5                   10                  15      


Asn Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg 
            20                  25                  30          


Gln Arg Xaa 
        35  


<210> 5
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 5
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 6
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 6
Pro Lys Pro Lys Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 7
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 7
Pro Lys Pro Glu Ala Pro Lys Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 8
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 8
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 9
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 9
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 10
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 10
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 11
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> Homotyrosine

<400> 11
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 12
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> D-Tyr

<400> 12
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 13
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 13
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 14
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (20)..(20)
<223> D-Lys

<400> 14
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Xaa Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 15
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (8)..(8)
<223> D-Lys

<400> 15
Pro Lys Pro Glu Ala Pro Gly Xaa Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 16
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 16
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 17
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 17
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 18
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (8)..(8)
<223> D-Lys

<400> 18
Pro Lys Pro Glu Ala Pro Gly Xaa Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 19
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 19
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 20
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 20
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 21
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (20)..(20)
<223> D-Lys

<400> 21
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Xaa Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 22
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (20)..(20)
<223> Dap

<400> 22
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Xaa Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 23
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 23
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Gln 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 24
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 24
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 25
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 25
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Ser 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 26
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 26
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Thr 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 27
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 27
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 28
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 28
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 29
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 29
Pro Lys Pro Glu Lys Pro Gly Glu Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 30
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (16)..(16)
<223> homoSer

<400> 30
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Xaa 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 31
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (16)..(16)
<223> alpha-methyl-Ser

<400> 31
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Xaa 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 32
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 32
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 33
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 33
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 34
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 34
Pro Lys Pro Glu Lys Pro Gly Glu Asp Ala Ser Pro Lys Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 35
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 35
Pro Lys Pro Glu Lys Pro Gly Glu Asp Ala Ser Pro Lys Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 36
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 36
Pro Lys Pro Glu Lys Pro Gly Glu Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 37
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 37
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 38
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 38
Pro Lys Pro Glu Lys Pro Gly Glu Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 39
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 39
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Glu 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 40
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 40
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 41
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 41
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Glu 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 42
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 42
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 43
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 43
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Glu Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 44
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 44
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Asp Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 45
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 45
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 46
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 46
Pro Lys Pro Glu Ala Pro Gly Lys Lys Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 47
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 47
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Asp Arg His Tyr Lys Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 48
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 48
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Lys Arg His Tyr Glu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 49
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> Beta-homo-Tyr

<400> 49
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 50
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 50
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Lys 
            20                  25                  30          


Arg Phe 
        


<210> 51
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 51
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Lys Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 52
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 52
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Lys Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 53
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 53
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Lys His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 54
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 54
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 55
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 55
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 56
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> 4-pyridylAla

<400> 56
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 57
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> 3-pyridylAla

<400> 57
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 58
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> 4-methylPhe

<400> 58
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 59
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> 4-carboxyPhe

<400> 59
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 60
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> 4-fluoroPhe

<400> 60
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 61
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> Homo-Phe

<400> 61
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 62
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylPhe

<400> 62
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 63
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylTyr

<400> 63
Pro Lys Pro Glu Ala Pro Lys Lys Asp Ala Ser Pro Glu Glu Leu Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 64
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 64
Pro Lys Pro Glu Ala Pro Lys Lys Asp Ala Ser Pro Glu Glu Leu Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 65
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (20)..(20)
<223> D-Lys

<400> 65
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Xaa Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 66
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 66
Pro Lys Pro Glu Ala Pro Gly Lys Asp Lys Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 67
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 67
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Lys Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 68
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 68
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Lys Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 69
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 69
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Lys Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 70
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 70
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 71
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 71
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 72
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 72
Pro Lys Pro Glu Lys Pro Gly Glu Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 73
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 73
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 74
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 74
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 75
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 75
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Ser 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 76
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 76
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 77
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 77
Pro Lys Pro Glu Lys Pro Gly Glu Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 78
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 78
Pro Lys Pro Glu Lys Pro Gly Glu Asp Ala Ser Pro Lys Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 79

<400> 79
000


<210> 80

<400> 80
000


<210> 81

<400> 81
000


<210> 82

<400> 82
000


<210> 83

<400> 83
000


<210> 84

<400> 84
000


<210> 85

<400> 85
000


<210> 86

<400> 86
000


<210> 87

<400> 87
000


<210> 88

<400> 88
000


<210> 89

<400> 89
000


<210> 90
<211> 35
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> VARIANT
<222> (1)..(1)
<223> /replace=" "

<220>
<221> VARIANT
<222> (5)..(5)
<223> /replace="K"

<220>
<221> VARIANT
<222> (6)..(6)
<223> /replace="K"

<220>
<221> VARIANT
<222> (8)..(8)
<223> /replace="K"

<220>
<221> VARIANT
<222> (9)..(9)
<223> /replace="K" or "k"

<220>
<221> VARIANT
<222> (10)..(10)
<223> /replace="K"

<220>
<221> VARIANT
<222> (11)..(11)
<223> /replace="K"

<220>
<221> VARIANT
<222> (14)..(14)
<223> /replace="K"

<220>
<221> VARIANT
<222> (15)..(15)
<223> /replace="K"

<220>
<221> VARIANT
<222> (16)..(16)
<223> /replace="W"

<220>
<221> VARIANT
<222> (17)..(17)
<223> /replace="E" or "K" or "N" or "Q" or "S" or "T" or 
      "alpha-methylserine" or "homoserine"

<220>
<221> VARIANT
<222> (19)..(19)
<223> /replace="Y"

<220>
<221> VARIANT
<222> (20)..(20)
<223> /replace="Y"

<220>
<221> VARIANT
<222> (21)..(21)
<223> /replace="D" or "E" or "K" or "k" or "Dap"

<220>
<221> VARIANT
<222> (23)..(23)
<223> /replace="D" or "K" or "L"

<220>
<221> VARIANT
<222> (24)..(24)
<223> /replace="R"

<220>
<221> VARIANT
<222> (26)..(26)
<223> /replace="Y"

<220>
<221> VARIANT
<222> (27)..(27)
<223> /replace="K" or "L"

<220>
<221> VARIANT
<222> (28)..(28)
<223> /replace="N"

<220>
<221> VARIANT
<222> (33)..(33)
<223> /replace="Q"

<220>
<221> VARIANT
<222> (35)..(35)
<223> /replace="y" or "3-pyridinylalanine" or "4-pyridinylalanine" or 
      "4-carboxyphenylalanine" or "4-fluorophenylalanine" or 
      "4-methylphenylalanine" or "N-methylphenylalanine" or 
      "homophenylalanine" or "beta-homotyrosine" or 

<220>
<221> VARIANT
<222> (35)..(35)
<223> CONT. FROM ABOVE: "homotyrosine" or "N-methyltyrosine"

<220>
<221> SITE
<222> (1)..(35)
<223> /note="Variant residues given in the sequence have no 
      preference with respect to those in the annotations 
      for variant positions"

<220> 
<221> source
<223> /note="See specification as filed for detailed description of
      substitutions and preferred embodiments"

<400> 90
Lys Pro Lys Pro Glu Ala Pro Gly Glu Asp Ala Ser Pro Glu Glu Leu 
1               5                   10                  15      


Asp Arg Lys Lys Ala Asp Ala Lys His Lys Glu Lys Trp Leu Thr Arg 
            20                  25                  30          


Lys Arg Phe 
        35  


<210> 91
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> VARIANT
<222> (5)..(5)
<223> /replace="K"

<220>
<221> VARIANT
<222> (7)..(7)
<223> /replace="K"

<220>
<221> VARIANT
<222> (8)..(8)
<223> /replace="K" or "k"

<220>
<221> VARIANT
<222> (13)..(13)
<223> /replace="K"

<220>
<221> VARIANT
<222> (15)..(15)
<223> /replace="W"

<220>
<221> VARIANT
<222> (16)..(16)
<223> /replace="E" or "K" or "N" or "S" or "alpha-methylserine" or 
      "homoserine"

<220>
<221> VARIANT
<222> (20)..(20)
<223> /replace="D" or "E" or "K" or "k"

<220>
<221> VARIANT
<222> (22)..(22)
<223> /replace="L"

<220>
<221> VARIANT
<222> (34)..(34)
<223> /replace="3-pyridinylalanine" or "4-pyridinylalanine" or 
      "4-carboxyphenylalanine" or "4-fluorophenylalanine" or 
      "4-methylphenylalanine" or "N-methylphenylalanine" or 
      "homophenylalanine" or "beta-homotyrosine" or 

<220>
<221> VARIANT
<222> (34)..(34)
<223> CONT. FROM ABOVE: "homotyrosine" or "N-methyltyrosine"

<220>
<221> SITE
<222> (1)..(34)
<223> /note="Variant residues given in the sequence have no 
      preference with respect to those in the annotations 
      for variant positions"

<220> 
<221> source
<223> /note="See specification as filed for detailed description of
      substitutions and preferred embodiments"

<400> 91
Pro Lys Pro Glu Ala Pro Gly Glu Asp Ala Ser Pro Glu Glu Leu Asp 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 92
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> VARIANT
<222> (5)..(5)
<223> /replace="K"

<220>
<221> VARIANT
<222> (7)..(7)
<223> /replace="K"

<220>
<221> VARIANT
<222> (8)..(8)
<223> /replace="K" or "k"

<220>
<221> VARIANT
<222> (13)..(13)
<223> /replace="K"

<220>
<221> VARIANT
<222> (15)..(15)
<223> /replace="W"

<220>
<221> VARIANT
<222> (16)..(16)
<223> /replace="E" or "K" or "S" or "alpha-methylserine" or 
      "homoserine"

<220>
<221> VARIANT
<222> (20)..(20)
<223> /replace="D" or "E" or "K" or "k"

<220>
<221> VARIANT
<222> (22)..(22)
<223> /replace="L"

<220>
<221> VARIANT
<222> (34)..(34)
<223> /replace="3-pyridinylalanine" or "4-pyridinylalanine" or 
      "4-carboxyphenylalanine" or "4-fluorophenylalanine" or 
      "4-methylphenylalanine" or "N-methylphenylalanine" or 
      "homophenylalanine" or "beta-homotyrosine" or 

<220>
<221> VARIANT
<222> (34)..(34)
<223> CONT. FROM ABOVE: "homotyrosine" or "N-methyltyrosine"

<220>
<221> SITE
<222> (1)..(34)
<223> /note="Variant residues given in the sequence have no 
      preference with respect to those in the annotations 
      for variant positions"

<220> 
<221> source
<223> /note="See specification as filed for detailed description of
      substitutions and preferred embodiments"

<400> 92
Pro Lys Pro Glu Ala Pro Gly Glu Asp Ala Ser Pro Glu Glu Leu Asp 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 93
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> VARIANT
<222> (5)..(5)
<223> /replace="K"

<220>
<221> VARIANT
<222> (7)..(7)
<223> /replace="K"

<220>
<221> VARIANT
<222> (8)..(8)
<223> /replace="K" or "k"

<220>
<221> VARIANT
<222> (13)..(13)
<223> /replace="K"

<220>
<221> VARIANT
<222> (15)..(15)
<223> /replace="W"

<220>
<221> VARIANT
<222> (16)..(16)
<223> /replace="E" or "K" or "N" or "S" or "alpha-methylserine" or 
      "homoserine"

<220>
<221> VARIANT
<222> (20)..(20)
<223> /replace="E" or "K" or "k"

<220>
<221> VARIANT
<222> (22)..(22)
<223> /replace="L"

<220>
<221> VARIANT
<222> (34)..(34)
<223> /replace="3-pyridinylalanine" or "4-pyridinylalanine" or 
      "4-carboxyphenylalanine" or "4-fluorophenylalanine" or 
      "4-methylphenylalanine" or "N-methylphenylalanine" or 
      "homophenylalanine" or "beta-homotyrosine" or 

<220>
<221> VARIANT
<222> (34)..(34)
<223> CONT. FROM ABOVE: "homotyrosine" or "N-methyltyrosine"

<220>
<221> SITE
<222> (1)..(34)
<223> /note="Variant residues given in the sequence have no 
      preference with respect to those in the annotations 
      for variant positions"

<220> 
<221> source
<223> /note="See specification as filed for detailed description of
      substitutions and preferred embodiments"

<400> 93
Pro Lys Pro Glu Ala Pro Gly Glu Asp Ala Ser Pro Glu Glu Leu Asp 
1               5                   10                  15      


Arg Tyr Tyr Asp Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 94
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> VARIANT
<222> (5)..(5)
<223> /replace="K"

<220>
<221> VARIANT
<222> (8)..(8)
<223> /replace="K" or "k"

<220>
<221> VARIANT
<222> (13)..(13)
<223> /replace="K"

<220>
<221> VARIANT
<222> (16)..(16)
<223> /replace="E" or "K" or "N"

<220>
<221> VARIANT
<222> (20)..(20)
<223> /replace="D" or "E" or "K" or "k"

<220>
<221> VARIANT
<222> (22)..(22)
<223> /replace="L"

<220>
<221> VARIANT
<222> (34)..(34)
<223> /replace="N-methyltyrosine"

<220>
<221> SITE
<222> (1)..(34)
<223> /note="Variant residues given in the sequence have no 
      preference with respect to those in the annotations 
      for variant positions"

<220> 
<221> source
<223> /note="See specification as filed for detailed description of
      substitutions and preferred embodiments"

<400> 94
Pro Lys Pro Glu Ala Pro Gly Glu Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 95
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> VARIANT
<222> (5)..(5)
<223> /replace="K"

<220>
<221> VARIANT
<222> (13)..(13)
<223> /replace="K"

<220>
<221> VARIANT
<222> (16)..(16)
<223> /replace="E" or "K" or "N"

<220>
<221> VARIANT
<222> (20)..(20)
<223> /replace="D" or "E" or "K" or "k"

<220>
<221> SITE
<222> (1)..(34)
<223> /note="Variant residues given in the sequence have no 
      preference with respect to those in the annotations 
      for variant positions"

<220> 
<221> source
<223> /note="See specification as filed for detailed description of
      substitutions and preferred embodiments"

<400> 95
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 96

<400> 96
000


<210> 97

<400> 97
000


<210> 98

<400> 98
000


<210> 99

<400> 99
000


<210> 100

<400> 100
000


<210> 101
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 101
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Tyr 
        


<210> 102

<400> 102
000


<210> 103

<400> 103
000


<210> 104
<211> 35
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (35)..(35)
<223> n-methylY

<400> 104
Lys Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp 
1               5                   10                  15      


Asn Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg 
            20                  25                  30          


Gln Arg Xaa 
        35  


<210> 105
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 105
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 106
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 106
Pro Lys Pro Lys Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 107
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 107
Pro Lys Pro Glu Ala Pro Lys Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 108
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 108
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 109
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 109
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 110
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylY

<400> 110
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 111
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> Homotyrosine

<400> 111
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 112
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> D-Tyr

<400> 112
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 113
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 113
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 114
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (20)..(20)
<223> D-Lys

<400> 114
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Xaa Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 115
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (8)..(8)
<223> D-Lys

<400> 115
Pro Lys Pro Glu Ala Pro Gly Xaa Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 116
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 116
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 117

<400> 117
000


<210> 118

<400> 118
000


<210> 119
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 119
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 120
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 120
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 121

<400> 121
000


<210> 122
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (20)..(20)
<223> Dap

<400> 122
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Xaa Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 123
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 123
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Gln 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 124
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 124
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 125
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 125
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Ser 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 126
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 126
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Thr 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 127
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 127
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 128

<400> 128
000


<210> 129
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 129
Pro Lys Pro Glu Lys Pro Gly Glu Asp Ala Ser Pro Lys Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 130
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (16)..(16)
<223> HomoSer

<400> 130
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Xaa 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 131
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (16)..(16)
<223> alpha-methyl-Ser

<400> 131
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Xaa 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 132

<400> 132
000


<210> 133

<400> 133
000


<210> 134
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 134
Pro Lys Pro Glu Lys Pro Gly Glu Asp Ala Ser Pro Lys Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 135

<400> 135
000


<210> 136

<400> 136
000


<210> 137

<400> 137
000


<210> 138

<400> 138
000


<210> 139
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 139
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Glu 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 140
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 140
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 141
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 141
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Glu 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 142

<400> 142
000


<210> 143
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 143
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Glu Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 144
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 144
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Asp Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 145
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 145
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 146
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 146
Pro Lys Pro Glu Ala Pro Gly Lys Lys Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 147
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 147
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Asp Arg His Tyr Lys Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 148
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 148
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Lys Arg His Tyr Glu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 149
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> Beta-homoTyr

<400> 149
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 150
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 150
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Lys 
            20                  25                  30          


Arg Phe 
        


<210> 151
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 151
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Lys Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 152
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 152
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Lys Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 153
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 153
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Lys His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 154

<400> 154
000


<210> 155
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 155
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 156
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> 4-pyridylAla

<400> 156
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 157
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> 3-pyridylAla

<400> 157
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 158
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> 4-methylPhe

<400> 158
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 159
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> 4-carboxyPhe

<400> 159
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 160
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> 4-fluoroPhe

<400> 160
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 161
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> homoPhe

<400> 161
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 162
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylPhe

<400> 162
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 163
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (34)..(34)
<223> n-methylTyr

<400> 163
Pro Lys Pro Glu Ala Pro Lys Lys Asp Ala Ser Pro Glu Glu Leu Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Xaa 
        


<210> 164
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 164
Pro Lys Pro Glu Ala Pro Lys Lys Asp Ala Ser Pro Glu Glu Leu Asn 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 165

<400> 165
000


<210> 166
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 166
Pro Lys Pro Glu Ala Pro Gly Lys Asp Lys Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 167
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 167
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Lys Trp Asn 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 168
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 168
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Lys Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 169
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 169
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asn 
1               5                   10                  15      


Arg Tyr Lys Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 170

<400> 170
000


<210> 171

<400> 171
000


<210> 172

<400> 172
000


<210> 173

<400> 173
000


<210> 174

<400> 174
000


<210> 175
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 175
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Ser 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 176

<400> 176
000


<210> 177
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 177
Pro Lys Pro Glu Lys Pro Gly Glu Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 178

<400> 178
000


<210> 179
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 179
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Tyr 
        


<210> 180
<211> 33
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 180
Pro Lys Pro Glu Ala Pro Gly Asp Ala Ser Pro Glu Glu Trp Asp Arg 
1               5                   10                  15      


Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln Arg 
            20                  25                  30          


Phe 
    


<210> 181
<211> 33
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 181
Pro Lys Pro Glu Ala Pro Gly Asp Ala Ser Pro Glu Glu Trp Lys Arg 
1               5                   10                  15      


Tyr Tyr Glu Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln Arg 
            20                  25                  30          


Phe 
    


<210> 182

<400> 182
000


<210> 183

<400> 183
000


<210> 184

<400> 184
000


<210> 185

<400> 185
000


<210> 186

<400> 186
000


<210> 187

<400> 187
000


<210> 188

<400> 188
000


<210> 189

<400> 189
000


<210> 190

<400> 190
000


<210> 191

<400> 191
000


<210> 192

<400> 192
000


<210> 193

<400> 193
000


<210> 194

<400> 194
000


<210> 195

<400> 195
000


<210> 196

<400> 196
000


<210> 197

<400> 197
000


<210> 198

<400> 198
000


<210> 199

<400> 199
000


<210> 200

<400> 200
000


<210> 201

<400> 201
000


<210> 202

<400> 202
000


<210> 203

<400> 203
000


<210> 204

<400> 204
000


<210> 205

<400> 205
000


<210> 206

<400> 206
000


<210> 207

<400> 207
000


<210> 208

<400> 208
000


<210> 209

<400> 209
000


<210> 210

<400> 210
000


<210> 211

<400> 211
000


<210> 212

<400> 212
000


<210> 213

<400> 213
000


<210> 214

<400> 214
000


<210> 215

<400> 215
000


<210> 216

<400> 216
000


<210> 217

<400> 217
000


<210> 218

<400> 218
000


<210> 219

<400> 219
000


<210> 220

<400> 220
000


<210> 221

<400> 221
000


<210> 222

<400> 222
000


<210> 223

<400> 223
000


<210> 224

<400> 224
000


<210> 225

<400> 225
000


<210> 226

<400> 226
000


<210> 227

<400> 227
000


<210> 228

<400> 228
000


<210> 229

<400> 229
000


<210> 230

<400> 230
000


<210> 231

<400> 231
000


<210> 232

<400> 232
000


<210> 233

<400> 233
000


<210> 234

<400> 234
000


<210> 235

<400> 235
000


<210> 236

<400> 236
000


<210> 237

<400> 237
000


<210> 238

<400> 238
000


<210> 239
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 239
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Glu 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 240
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 240
Pro Lys Pro Glu Lys Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 241
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 241
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Glu 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 242
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 242
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 243
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 243
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Glu Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 244
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 244
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Asp Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 245
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 245
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Lys Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 246
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 246
Pro Lys Pro Glu Ala Pro Gly Lys Lys Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 247
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 247
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Asp Arg His Tyr Lys Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 248
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 248
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Lys Arg His Tyr Glu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 249

<400> 249
000


<210> 250

<400> 250
000


<210> 251

<400> 251
000


<210> 252

<400> 252
000


<210> 253

<400> 253
000


<210> 254

<400> 254
000


<210> 255

<400> 255
000


<210> 256

<400> 256
000


<210> 257

<400> 257
000


<210> 258

<400> 258
000


<210> 259

<400> 259
000


<210> 260

<400> 260
000


<210> 261

<400> 261
000


<210> 262

<400> 262
000


<210> 263

<400> 263
000


<210> 264

<400> 264
000


<210> 265

<400> 265
000


<210> 266

<400> 266
000


<210> 267

<400> 267
000


<210> 268

<400> 268
000


<210> 269

<400> 269
000


<210> 270

<400> 270
000


<210> 271

<400> 271
000


<210> 272

<400> 272
000


<210> 273

<400> 273
000


<210> 274

<400> 274
000


<210> 275

<400> 275
000


<210> 276

<400> 276
000


<210> 277

<400> 277
000


<210> 278

<400> 278
000


<210> 279

<400> 279
000


<210> 280
<211> 33
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 280
Pro Lys Pro Glu Ala Pro Gly Asp Ala Ser Pro Glu Glu Trp Asp Arg 
1               5                   10                  15      


Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln Arg 
            20                  25                  30          


Phe 
    


<210> 281
<211> 33
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 281
Pro Lys Pro Glu Ala Pro Gly Asp Ala Ser Pro Glu Glu Trp Lys Arg 
1               5                   10                  15      


Tyr Tyr Glu Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln Arg 
            20                  25                  30          


Phe 
    


<210> 282

<400> 282
000


<210> 283

<400> 283
000


<210> 284

<400> 284
000


<210> 285

<400> 285
000


<210> 286

<400> 286
000


<210> 287

<400> 287
000


<210> 288

<400> 288
000


<210> 289

<400> 289
000


<210> 290

<400> 290
000


<210> 291

<400> 291
000


<210> 292

<400> 292
000


<210> 293

<400> 293
000


<210> 294

<400> 294
000


<210> 295

<400> 295
000


<210> 296

<400> 296
000


<210> 297

<400> 297
000


<210> 298

<400> 298
000


<210> 299

<400> 299
000


<210> 300

<400> 300
000


<210> 301

<400> 301
000


<210> 302

<400> 302
000


<210> 303

<400> 303
000


<210> 304

<400> 304
000


<210> 305

<400> 305
000


<210> 306

<400> 306
000


<210> 307

<400> 307
000


<210> 308

<400> 308
000


<210> 309

<400> 309
000


<210> 310

<400> 310
000


<210> 311

<400> 311
000


<210> 312

<400> 312
000


<210> 313

<400> 313
000


<210> 314

<400> 314
000


<210> 315

<400> 315
000


<210> 316

<400> 316
000


<210> 317

<400> 317
000


<210> 318

<400> 318
000


<210> 319

<400> 319
000


<210> 320

<400> 320
000


<210> 321

<400> 321
000


<210> 322

<400> 322
000


<210> 323

<400> 323
000


<210> 324
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 324
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 325

<400> 325
000


<210> 326

<400> 326
000


<210> 327

<400> 327
000


<210> 328

<400> 328
000


<210> 329

<400> 329
000


<210> 330

<400> 330
000


<210> 331

<400> 331
000


<210> 332

<400> 332
000


<210> 333

<400> 333
000


<210> 334

<400> 334
000


<210> 335

<400> 335
000


<210> 336

<400> 336
000


<210> 337

<400> 337
000


<210> 338

<400> 338
000


<210> 339

<400> 339
000


<210> 340

<400> 340
000


<210> 341

<400> 341
000


<210> 342
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 342
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 343
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 343
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Glu Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 344

<400> 344
000


<210> 345

<400> 345
000


<210> 346

<400> 346
000


<210> 347

<400> 347
000


<210> 348

<400> 348
000


<210> 349

<400> 349
000


<210> 350

<400> 350
000


<210> 351

<400> 351
000


<210> 352

<400> 352
000


<210> 353

<400> 353
000


<210> 354

<400> 354
000


<210> 355

<400> 355
000


<210> 356

<400> 356
000


<210> 357

<400> 357
000


<210> 358

<400> 358
000


<210> 359

<400> 359
000


<210> 360

<400> 360
000


<210> 361

<400> 361
000


<210> 362

<400> 362
000


<210> 363

<400> 363
000


<210> 364

<400> 364
000


<210> 365

<400> 365
000


<210> 366

<400> 366
000


<210> 367

<400> 367
000


<210> 368

<400> 368
000


<210> 369

<400> 369
000


<210> 370

<400> 370
000


<210> 371

<400> 371
000


<210> 372

<400> 372
000


<210> 373

<400> 373
000


<210> 374

<400> 374
000


<210> 375

<400> 375
000


<210> 376

<400> 376
000


<210> 377

<400> 377
000


<210> 378

<400> 378
000


<210> 379

<400> 379
000


<210> 380

<400> 380
000


<210> 381

<400> 381
000


<210> 382

<400> 382
000


<210> 383

<400> 383
000


<210> 384

<400> 384
000


<210> 385

<400> 385
000


<210> 386

<400> 386
000


<210> 387

<400> 387
000


<210> 388

<400> 388
000


<210> 389

<400> 389
000


<210> 390
<211> 35
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> VARIANT
<222> (1)..(1)
<223> /replace=" "

<220>
<221> VARIANT
<222> (5)..(5)
<223> /replace="K"

<220>
<221> VARIANT
<222> (6)..(6)
<223> /replace="K"

<220>
<221> VARIANT
<222> (8)..(8)
<223> /replace="K"

<220>
<221> VARIANT
<222> (9)..(9)
<223> /replace="K" or "k"

<220>
<221> VARIANT
<222> (10)..(10)
<223> /replace="K"

<220>
<221> VARIANT
<222> (11)..(11)
<223> /replace="K"

<220>
<221> VARIANT
<222> (14)..(14)
<223> /replace="K"

<220>
<221> VARIANT
<222> (15)..(15)
<223> /replace="K"

<220>
<221> VARIANT
<222> (16)..(16)
<223> /replace="W"

<220>
<221> VARIANT
<222> (17)..(17)
<223> /replace="E" or "K" or "N" or "Q" or "S" or "T" or 
      "alpha-methylserine" or "homoserine"

<220>
<221> VARIANT
<222> (19)..(19)
<223> /replace="Y"

<220>
<221> VARIANT
<222> (20)..(20)
<223> /replace="Y"

<220>
<221> VARIANT
<222> (21)..(21)
<223> /replace="D" or "E" or "K" or "k" or "Dap"

<220>
<221> VARIANT
<222> (23)..(23)
<223> /replace="D" or "K" or "L"

<220>
<221> VARIANT
<222> (24)..(24)
<223> /replace="R"

<220>
<221> VARIANT
<222> (26)..(26)
<223> /replace="Y"

<220>
<221> VARIANT
<222> (27)..(27)
<223> /replace="K" or "L"

<220>
<221> VARIANT
<222> (28)..(28)
<223> /replace="N"

<220>
<221> VARIANT
<222> (33)..(33)
<223> /replace="Q"

<220>
<221> VARIANT
<222> (35)..(35)
<223> /replace="y" or "3-pyridinylalanine" or "4-pyridinylalanine" or 
      "4-carboxyphenylalanine" or "4-fluorophenylalanine" or 
      "4-methylphenylalanine" or "N-methylphenylalanine" or 
      "homophenylalanine" or "beta-homotyrosine" or 

<220>
<221> VARIANT
<222> (35)..(35)
<223> CONT. FROM ABOVE: "homotyrosine" or "N-methyltyrosine"

<220>
<221> SITE
<222> (1)..(35)
<223> /note="Variant residues given in the sequence have no 
      preference with respect to those in the annotations 
      for variant positions"

<220> 
<221> source
<223> /note="See specification as filed for detailed description of
      substitutions and preferred embodiments"

<400> 390
Lys Pro Lys Pro Glu Ala Pro Gly Glu Asp Ala Ser Pro Glu Glu Leu 
1               5                   10                  15      


Asp Arg Lys Lys Ala Asp Ala Lys His Lys Glu Lys Trp Leu Thr Arg 
            20                  25                  30          


Lys Arg Phe 
        35  


<210> 391

<400> 391
000


<210> 392

<400> 392
000


<210> 393

<400> 393
000


<210> 394
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> VARIANT
<222> (5)..(5)
<223> /replace="K"

<220>
<221> VARIANT
<222> (8)..(8)
<223> /replace="K" or "k"

<220>
<221> VARIANT
<222> (13)..(13)
<223> /replace="K"

<220>
<221> VARIANT
<222> (16)..(16)
<223> /replace="E" or "K" or "N"

<220>
<221> VARIANT
<222> (20)..(20)
<223> /replace="D" or "E" or "K" or "k"

<220>
<221> VARIANT
<222> (22)..(22)
<223> /replace="L"

<220>
<221> VARIANT
<222> (34)..(34)
<223> /replace="N-methyltyrosine"

<220>
<221> SITE
<222> (1)..(34)
<223> /note="Variant residues given in the sequence have no 
      preference with respect to those in the annotations 
      for variant positions"

<220> 
<221> source
<223> /note="See specification as filed for detailed description of
      substitutions and preferred embodiments"

<400> 394
Pro Lys Pro Glu Ala Pro Gly Glu Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Ala Asp Ala Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 395

<400> 395
000


<210> 396

<400> 396
000


<210> 397

<400> 397
000


<210> 398

<400> 398
000


<210> 399

<400> 399
000


<210> 400

<400> 400
000


<210> 401

<400> 401
000


<210> 402

<400> 402
000


<210> 403

<400> 403
000


<210> 404

<400> 404
000


<210> 405

<400> 405
000


<210> 406

<400> 406
000


<210> 407

<400> 407
000


<210> 408

<400> 408
000


<210> 409

<400> 409
000


<210> 410

<400> 410
000


<210> 411

<400> 411
000


<210> 412

<400> 412
000


<210> 413

<400> 413
000


<210> 414

<400> 414
000


<210> 415

<400> 415
000


<210> 416

<400> 416
000


<210> 417

<400> 417
000


<210> 418

<400> 418
000


<210> 419

<400> 419
000


<210> 420

<400> 420
000


<210> 421

<400> 421
000


<210> 422

<400> 422
000


<210> 423

<400> 423
000


<210> 424
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 424
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 425

<400> 425
000


<210> 426

<400> 426
000


<210> 427

<400> 427
000


<210> 428

<400> 428
000


<210> 429

<400> 429
000


<210> 430

<400> 430
000


<210> 431

<400> 431
000


<210> 432

<400> 432
000


<210> 433

<400> 433
000


<210> 434

<400> 434
000


<210> 435

<400> 435
000


<210> 436

<400> 436
000


<210> 437

<400> 437
000


<210> 438

<400> 438
000


<210> 439

<400> 439
000


<210> 440

<400> 440
000


<210> 441

<400> 441
000


<210> 442
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 442
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 443
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"

<400> 443
Pro Lys Pro Glu Ala Pro Gly Lys Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Glu Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 444

<400> 444
000


<210> 445

<400> 445
000


<210> 446

<400> 446
000


<210> 447

<400> 447
000


<210> 448

<400> 448
000


<210> 449

<400> 449
000


<210> 450

<400> 450
000


<210> 451

<400> 451
000


<210> 452

<400> 452
000


<210> 453

<400> 453
000


<210> 454

<400> 454
000


<210> 455

<400> 455
000


<210> 456

<400> 456
000


<210> 457

<400> 457
000


<210> 458

<400> 458
000


<210> 459

<400> 459
000


<210> 460

<400> 460
000


<210> 461

<400> 461
000


<210> 462

<400> 462
000


<210> 463

<400> 463
000


<210> 464

<400> 464
000


<210> 465

<400> 465
000


<210> 466

<400> 466
000


<210> 467

<400> 467
000


<210> 468

<400> 468
000


<210> 469

<400> 469
000


<210> 470

<400> 470
000


<210> 471

<400> 471
000


<210> 472

<400> 472
000


<210> 473

<400> 473
000


<210> 474

<400> 474
000


<210> 475

<400> 475
000


<210> 476

<400> 476
000


<210> 477

<400> 477
000


<210> 478

<400> 478
000


<210> 479

<400> 479
000


<210> 480

<400> 480
000


<210> 481

<400> 481
000


<210> 482

<400> 482
000


<210> 483

<400> 483
000


<210> 484

<400> 484
000


<210> 485

<400> 485
000


<210> 486

<400> 486
000


<210> 487

<400> 487
000


<210> 488

<400> 488
000


<210> 489

<400> 489
000


<210> 490

<400> 490
000


<210> 491

<400> 491
000


<210> 492

<400> 492
000


<210> 493

<400> 493
000


<210> 494

<400> 494
000


<210> 495

<400> 495
000


<210> 496

<400> 496
000


<210> 497

<400> 497
000


<210> 498

<400> 498
000


<210> 499

<400> 499
000


<210> 500

<400> 500
000


<210> 501

<400> 501
000


<210> 502

<400> 502
000


<210> 503

<400> 503
000


<210> 504

<400> 504
000


<210> 505

<400> 505
000


<210> 506

<400> 506
000


<210> 507

<400> 507
000


<210> 508

<400> 508
000


<210> 509

<400> 509
000


<210> 510

<400> 510
000


<210> 511

<400> 511
000


<210> 512

<400> 512
000


<210> 513

<400> 513
000


<210> 514

<400> 514
000


<210> 515

<400> 515
000


<210> 516

<400> 516
000


<210> 517

<400> 517
000


<210> 518

<400> 518
000


<210> 519

<400> 519
000


<210> 520

<400> 520
000


<210> 521

<400> 521
000


<210> 522

<400> 522
000


<210> 523

<400> 523
000


<210> 524
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (8)..(8)
<223> K(alloc)

<400> 524
Pro Lys Pro Glu Ala Pro Gly Xaa Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 525

<400> 525
000


<210> 526

<400> 526
000


<210> 527

<400> 527
000


<210> 528

<400> 528
000


<210> 529

<400> 529
000


<210> 530

<400> 530
000


<210> 531

<400> 531
000


<210> 532

<400> 532
000


<210> 533

<400> 533
000


<210> 534

<400> 534
000


<210> 535

<400> 535
000


<210> 536

<400> 536
000


<210> 537

<400> 537
000


<210> 538

<400> 538
000


<210> 539

<400> 539
000


<210> 540

<400> 540
000


<210> 541

<400> 541
000


<210> 542
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (8)..(8)
<223> K(ivDde)

<400> 542
Pro Lys Pro Glu Ala Pro Gly Xaa Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 543
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (8)..(8)
<223> K(ivDde)

<400> 543
Pro Lys Pro Glu Ala Pro Gly Xaa Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Glu Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 544

<400> 544
000


<210> 545

<400> 545
000


<210> 546

<400> 546
000


<210> 547

<400> 547
000


<210> 548

<400> 548
000


<210> 549

<400> 549
000


<210> 550

<400> 550
000


<210> 551

<400> 551
000


<210> 552

<400> 552
000


<210> 553

<400> 553
000


<210> 554

<400> 554
000


<210> 555

<400> 555
000


<210> 556

<400> 556
000


<210> 557

<400> 557
000


<210> 558

<400> 558
000


<210> 559

<400> 559
000


<210> 560

<400> 560
000


<210> 561

<400> 561
000


<210> 562

<400> 562
000


<210> 563

<400> 563
000


<210> 564

<400> 564
000


<210> 565

<400> 565
000


<210> 566

<400> 566
000


<210> 567

<400> 567
000


<210> 568

<400> 568
000


<210> 569

<400> 569
000


<210> 570

<400> 570
000


<210> 571

<400> 571
000


<210> 572

<400> 572
000


<210> 573

<400> 573
000


<210> 574

<400> 574
000


<210> 575

<400> 575
000


<210> 576

<400> 576
000


<210> 577

<400> 577
000


<210> 578

<400> 578
000


<210> 579

<400> 579
000


<210> 580

<400> 580
000


<210> 581

<400> 581
000


<210> 582

<400> 582
000


<210> 583

<400> 583
000


<210> 584

<400> 584
000


<210> 585

<400> 585
000


<210> 586

<400> 586
000


<210> 587

<400> 587
000


<210> 588

<400> 588
000


<210> 589

<400> 589
000


<210> 590

<400> 590
000


<210> 591

<400> 591
000


<210> 592

<400> 592
000


<210> 593

<400> 593
000


<210> 594

<400> 594
000


<210> 595

<400> 595
000


<210> 596

<400> 596
000


<210> 597

<400> 597
000


<210> 598

<400> 598
000


<210> 599

<400> 599
000


<210> 600

<400> 600
000


<210> 601

<400> 601
000


<210> 602

<400> 602
000


<210> 603

<400> 603
000


<210> 604

<400> 604
000


<210> 605

<400> 605
000


<210> 606

<400> 606
000


<210> 607

<400> 607
000


<210> 608

<400> 608
000


<210> 609

<400> 609
000


<210> 610

<400> 610
000


<210> 611

<400> 611
000


<210> 612

<400> 612
000


<210> 613

<400> 613
000


<210> 614

<400> 614
000


<210> 615

<400> 615
000


<210> 616

<400> 616
000


<210> 617

<400> 617
000


<210> 618

<400> 618
000


<210> 619

<400> 619
000


<210> 620

<400> 620
000


<210> 621

<400> 621
000


<210> 622

<400> 622
000


<210> 623

<400> 623
000


<210> 624

<400> 624
000


<210> 625

<400> 625
000


<210> 626

<400> 626
000


<210> 627

<400> 627
000


<210> 628

<400> 628
000


<210> 629

<400> 629
000


<210> 630

<400> 630
000


<210> 631

<400> 631
000


<210> 632

<400> 632
000


<210> 633

<400> 633
000


<210> 634

<400> 634
000


<210> 635

<400> 635
000


<210> 636

<400> 636
000


<210> 637

<400> 637
000


<210> 638

<400> 638
000


<210> 639

<400> 639
000


<210> 640

<400> 640
000


<210> 641

<400> 641
000


<210> 642
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (8)..(8)
<223> K(ivDde)

<400> 642
Pro Lys Pro Glu Ala Pro Gly Xaa Asp Ala Ser Pro Glu Glu Trp Asp 
1               5                   10                  15      


Arg Tyr Tyr Lys Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 643
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (8)..(8)
<223> K(ivDde)

<400> 643
Pro Lys Pro Glu Ala Pro Gly Xaa Asp Ala Ser Pro Glu Glu Trp Lys 
1               5                   10                  15      


Arg Tyr Tyr Glu Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 644

<400> 644
000


<210> 645

<400> 645
000


<210> 646

<400> 646
000


<210> 647

<400> 647
000


<210> 648

<400> 648
000


<210> 649

<400> 649
000


<210> 650

<400> 650
000


<210> 651

<400> 651
000


<210> 652

<400> 652
000


<210> 653

<400> 653
000


<210> 654

<400> 654
000


<210> 655

<400> 655
000


<210> 656

<400> 656
000


<210> 657

<400> 657
000


<210> 658

<400> 658
000


<210> 659

<400> 659
000


<210> 660

<400> 660
000


<210> 661

<400> 661
000


<210> 662

<400> 662
000


<210> 663

<400> 663
000


<210> 664

<400> 664
000


<210> 665

<400> 665
000


<210> 666

<400> 666
000


<210> 667

<400> 667
000


<210> 668

<400> 668
000


<210> 669

<400> 669
000


<210> 670

<400> 670
000


<210> 671

<400> 671
000


<210> 672

<400> 672
000


<210> 673

<400> 673
000


<210> 674

<400> 674
000


<210> 675

<400> 675
000


<210> 676

<400> 676
000


<210> 677

<400> 677
000


<210> 678

<400> 678
000


<210> 679

<400> 679
000


<210> 680

<400> 680
000


<210> 681

<400> 681
000


<210> 682

<400> 682
000


<210> 683

<400> 683
000


<210> 684

<400> 684
000


<210> 685

<400> 685
000


<210> 686

<400> 686
000


<210> 687

<400> 687
000


<210> 688

<400> 688
000


<210> 689

<400> 689
000


<210> 690

<400> 690
000


<210> 691

<400> 691
000


<210> 692

<400> 692
000


<210> 693

<400> 693
000


<210> 694

<400> 694
000


<210> 695

<400> 695
000


<210> 696

<400> 696
000


<210> 697

<400> 697
000


<210> 698

<400> 698
000


<210> 699

<400> 699
000


<210> 700

<400> 700
000


<210> 701

<400> 701
000


<210> 702

<400> 702
000


<210> 703

<400> 703
000


<210> 704

<400> 704
000


<210> 705

<400> 705
000


<210> 706

<400> 706
000


<210> 707

<400> 707
000


<210> 708

<400> 708
000


<210> 709

<400> 709
000


<210> 710

<400> 710
000


<210> 711

<400> 711
000


<210> 712

<400> 712
000


<210> 713

<400> 713
000


<210> 714

<400> 714
000


<210> 715

<400> 715
000


<210> 716

<400> 716
000


<210> 717

<400> 717
000


<210> 718

<400> 718
000


<210> 719

<400> 719
000


<210> 720

<400> 720
000


<210> 721

<400> 721
000


<210> 722

<400> 722
000


<210> 723

<400> 723
000


<210> 724

<400> 724
000


<210> 725

<400> 725
000


<210> 726

<400> 726
000


<210> 727

<400> 727
000


<210> 728

<400> 728
000


<210> 729

<400> 729
000


<210> 730

<400> 730
000


<210> 731

<400> 731
000


<210> 732

<400> 732
000


<210> 733

<400> 733
000


<210> 734

<400> 734
000


<210> 735

<400> 735
000


<210> 736

<400> 736
000


<210> 737

<400> 737
000


<210> 738

<400> 738
000


<210> 739

<400> 739
000


<210> 740

<400> 740
000


<210> 741

<400> 741
000


<210> 742
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (8)..(8)
<223> K(ivDde)

<220>
<221> MOD_RES
<222> (16)..(16)
<223> D(allyl)

<220>
<221> MOD_RES
<222> (20)..(20)
<223> K(alloc)

<400> 742
Pro Lys Pro Glu Ala Pro Gly Xaa Asp Ala Ser Pro Glu Glu Trp Xaa 
1               5                   10                  15      


Arg Tyr Tyr Xaa Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 743
<211> 34
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (8)..(8)
<223> K(ivDde)

<220>
<221> MOD_RES
<222> (16)..(16)
<223> K(alloc)

<220>
<221> MOD_RES
<222> (20)..(20)
<223> E(allyl)

<400> 743
Pro Lys Pro Glu Ala Pro Gly Xaa Asp Ala Ser Pro Glu Glu Trp Xaa 
1               5                   10                  15      


Arg Tyr Tyr Xaa Asp Leu Arg His Tyr Leu Asn Trp Leu Thr Arg Gln 
            20                  25                  30          


Arg Phe 
        


<210> 744

<400> 744
000


<210> 745

<400> 745
000


<210> 746

<400> 746
000


<210> 747

<400> 747
000


<210> 748

<400> 748
000


<210> 749

<400> 749
000


<210> 750

<400> 750
000


<210> 751

<400> 751
000


<210> 752

<400> 752
000


<210> 753

<400> 753
000


<210> 754

<400> 754
000


<210> 755

<400> 755
000


<210> 756

<400> 756
000


<210> 757

<400> 757
000


<210> 758

<400> 758
000


<210> 759

<400> 759
000


<210> 760

<400> 760
000


<210> 761

<400> 761
000


<210> 762

<400> 762
000


<210> 763

<400> 763
000


<210> 764

<400> 764
000


<210> 765

<400> 765
000


<210> 766

<400> 766
000


<210> 767

<400> 767
000


<210> 768

<400> 768
000


<210> 769

<400> 769
000


<210> 770

<400> 770
000


<210> 771

<400> 771
000


<210> 772

<400> 772
000


<210> 773

<400> 773
000


<210> 774

<400> 774
000


<210> 775

<400> 775
000


<210> 776

<400> 776
000


<210> 777

<400> 777
000


<210> 778

<400> 778
000


<210> 779

<400> 779
000


<210> 780

<400> 780
000


<210> 781

<400> 781
000


<210> 782

<400> 782
000


<210> 783

<400> 783
000


<210> 784

<400> 784
000


<210> 785

<400> 785
000


<210> 786

<400> 786
000


<210> 787

<400> 787
000


<210> 788

<400> 788
000


<210> 789

<400> 789
000


<210> 790

<400> 790
000


<210> 791

<400> 791
000


<210> 792

<400> 792
000


<210> 793

<400> 793
000


<210> 794

<400> 794
000


<210> 795

<400> 795
000


<210> 796

<400> 796
000


<210> 797

<400> 797
000


<210> 798

<400> 798
000


<210> 799

<400> 799
000


<210> 800
<211> 36
<212> PRT
<213> Unknown

<220>
<221> source
<223> /note="Description of Unknown: 
      PYY peptide sequence"

<400> 800
Tyr Pro Ile Lys Pro Glu Ala Pro Gly Glu Asp Ala Ser Pro Glu Glu 
1               5                   10                  15      


Leu Asn Arg Tyr Tyr Ala Ser Leu Arg His Tyr Leu Asn Leu Val Thr 
            20                  25                  30          


Arg Gln Arg Tyr 
        35      


<210> 801
<211> 30
<212> PRT
<213> Unknown

<220>
<221> source
<223> /note="Description of Unknown: 
      GLP-1 sequence"

<400> 801
His Ala Glu Gly Thr Phe Thr Ser Asp Val Ser Ser Tyr Leu Glu Gly 
1               5                   10                  15      


Gln Ala Ala Lys Glu Phe Ile Ala Trp Leu Val Lys Gly Arg 
            20                  25                  30  


<210> 802
<211> 39
<212> PRT
<213> Unknown

<220>
<221> source
<223> /note="Description of Unknown: 
      Exenatide sequence"

<400> 802
His Gly Glu Gly Thr Phe Thr Ser Asp Leu Ser Lys Gln Met Glu Glu 
1               5                   10                  15      


Glu Ala Val Arg Leu Phe Ile Glu Trp Leu Lys Asn Gly Gly Pro Ser 
            20                  25                  30          


Ser Gly Ala Pro Pro Pro Ser 
        35                  


<210> 803

<400> 803
000


<210> 804

<400> 804
000


<210> 805
<211> 40
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> MOD_RES
<222> (2)..(2)
<223> Aib

<220>
<221> MOD_RES
<222> (13)..(13)
<223> Aib

<220>
<221> MOD_RES
<222> (20)..(20)
<223> diacid-gamma-Glu

<220>
<221> MOD_RES
<222> (21)..(21)
<223> (AEEA)2-Lys

<400> 805
Tyr Xaa Glu Gly Thr Phe Thr Ser Asp Tyr Ser Ile Xaa Leu Asp Lys 
1               5                   10                  15      


Ile Ala Gln Xaa Xaa Ala Phe Val Gln Trp Leu Ile Ala Gly Gly Pro 
            20                  25                  30          


Ser Ser Gly Ala Pro Pro Pro Ser 
        35                  40  


<210> 806
<211> 35
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      polypeptide"


<220>
<221> VARIANT
<222> (1)..(1)
<223> /replace=" "

<220>
<221> VARIANT
<222> (5)..(5)
<223> /replace="K"

<220>
<221> VARIANT
<222> (6)..(6)
<223> /replace="K"

<220>
<221> VARIANT
<222> (8)..(8)
<223> /replace="K"

<220>
<221> VARIANT
<222> (9)..(9)
<223> /replace="K" or "k"

<220>
<221> VARIANT
<222> (11)..(11)
<223> /replace="K"

<220>
<221> VARIANT
<222> (14)..(14)
<223> /replace="K"

<220>
<221> VARIANT
<222> (15)..(15)
<223> /replace="K"

<220>
<221> VARIANT
<222> (16)..(16)
<223> /replace="W"

<220>
<221> VARIANT
<222> (17)..(17)
<223> /replace="E" or "K" or "N" or "Q" or "S" or "T" or 
      "alpha-methylserine" or "homoserine"

<220>
<221> VARIANT
<222> (19)..(19)
<223> /replace="Y"

<220>
<221> VARIANT
<222> (20)..(20)
<223> /replace="Y"

<220>
<221> VARIANT
<222> (21)..(21)
<223> /replace="D" or "E" or "K" or "k" or "Dap"

<220>
<221> VARIANT
<222> (23)..(23)
<223> /replace="D" or "K" or "L"

<220>
<221> VARIANT
<222> (24)..(24)
<223> /replace="R"

<220>
<221> VARIANT
<222> (26)..(26)
<223> /replace="Y"

<220>
<221> VARIANT
<222> (28)..(28)
<223> /replace="N"

<220>
<221> VARIANT
<222> (33)..(33)
<223> /replace="Q"

<220>
<221> VARIANT
<222> (35)..(35)
<223> /replace="y" or "3-pyridinylalanine" or "4-pyridinylalanine" or 
      "4-carboxyphenylalanine" or "4-fluorophenylalanine" or 
      "4-methylphenylalanine" or "N-methylphenylalanine" or 
      "homophenylalanine" or "beta-homotyrosine" or 

<220>
<221> VARIANT
<222> (35)..(35)
<223> CONT. FROM ABOVE: "homotyrosine" or "N-methyltyrosine"

<220> 
<221> source
<223> /note="See specification as filed for detailed description of
      substitutions and preferred embodiments"

<400> 806
Lys Pro Lys Pro Glu Ala Pro Gly Glu Asp Ala Ser Pro Glu Glu Leu 
1               5                   10                  15      


Asp Arg Lys Lys Ala Asp Ala Lys His Lys Leu Lys Trp Leu Thr Arg 
            20                  25                  30          


Lys Arg Phe 
        35  


<210> 807
<211> 7
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      peptide"

<400> 807
Trp Asp Arg Tyr Tyr Lys Asp 
1               5           


<210> 808
<211> 10
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      peptide"


<220>
<221> MOD_RES
<222> (1)..(10)
<223> Gamma-Glu

<220>
<221> SITE
<222> (1)..(10)
<223> /note="This sequence may encompass 1-10 residues"

<400> 808
Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa 
1               5                   10  


<210> 809
<211> 11
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      peptide"


<220>
<221> MOD_RES
<222> (1)..(10)
<223> Gamma-Glu

<220>
<221> SITE
<222> (1)..(10)
<223> /note="This sequence may encompass 1-10 'Xaa' residues"

<400> 809
Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Gly 
1               5                   10      


<210> 810
<211> 4
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      peptide"


<220>
<221> MOD_RES
<222> (1)..(4)
<223> Gamma-Glu

<400> 810
Xaa Xaa Xaa Xaa 
1               


<210> 811
<211> 5
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      peptide"


<220>
<221> MOD_RES
<222> (1)..(5)
<223> Gamma-Glu

<400> 811
Xaa Xaa Xaa Xaa Xaa 
1               5   


<210> 812
<211> 4
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      peptide"


<220>
<221> MOD_RES
<222> (1)..(3)
<223> Gamma-Glu

<400> 812
Xaa Xaa Xaa Gly 
1               


<210> 813
<211> 11
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      peptide"


<220>
<221> MOD_RES
<222> (2)..(11)
<223> Gamma-Glu

<220>
<221> SITE
<222> (2)..(11)
<223> /note="This sequence may encompass 1-10 'Xaa' residues"

<400> 813
Gly Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa 
1               5                   10      


<210> 814
<211> 4
<212> PRT
<213> Artificial Sequence

<220>
<221> source
<223> /note="Description of Artificial Sequence: Synthetic
      peptide"

<400> 814
Glu Glu Glu Glu 
1               
