                         SEQUENCE LISTING

<110>  Synaffix B.V.
 
<120>  DAR1 conjugates via cycloaddition

<130>  P6090977PCT

<150>  EP 20151551.7
<151>  2020-01-13

<160>  6     

<170>  PatentIn version 3.5

<210>  1
<211>  26
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Sequence identification of C-terminal sortase A recognition 
       sequence

<400>  1

Gly Gly Gly Gly Ser Gly Gly Gly Gly Ser Leu Pro Glu Thr Gly Gly 
1               5                   10                  15      


His His His His His His His His His His 
            20                  25      


<210>  2
<211>  192
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Sequence identification of sortase A

<400>  2

Thr Gly Ser His His His His His His Gly Ser Lys Pro His Ile Asp 
1               5                   10                  15      


Asn Tyr Leu His Asp Lys Asp Lys Asp Glu Lys Ile Glu Gln Tyr Asp 
            20                  25                  30          


Lys Asn Val Lys Glu Gln Ala Ser Lys Asp Lys Lys Gln Gln Ala Lys 
        35                  40                  45              


Pro Gln Ile Pro Lys Asp Lys Ser Lys Val Ala Gly Tyr Ile Glu Ile 
    50                  55                  60                  


Pro Asp Ala Asp Ile Lys Glu Pro Val Tyr Pro Gly Pro Ala Thr Pro 
65                  70                  75                  80  


Glu Gln Leu Asn Arg Gly Val Ser Phe Ala Glu Glu Asn Glu Ser Leu 
                85                  90                  95      


Asp Asp Gln Asn Ile Ser Ile Ala Gly His Thr Phe Ile Asp Arg Pro 
            100                 105                 110         


Asn Tyr Gln Phe Thr Asn Leu Lys Ala Ala Lys Lys Gly Ser Met Val 
        115                 120                 125             


Tyr Phe Lys Val Gly Asn Glu Thr Arg Lys Tyr Lys Met Thr Ser Ile 
    130                 135                 140                 


Arg Asp Val Lys Pro Thr Asp Val Gly Val Leu Asp Glu Gln Lys Gly 
145                 150                 155                 160 


Lys Asp Lys Gln Leu Thr Leu Ile Thr Cys Asp Asp Tyr Asn Glu Lys 
                165                 170                 175     


Thr Gly Val Trp Glu Lys Arg Lys Ile Phe Val Ala Thr Glu Val Lys 
            180                 185                 190         


<210>  3
<211>  233
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Sequence identification of His6-TEVsite-GGG-IL15R -IL15

<400>  3

Met Gly Ser Ser His His His His His His Ser Ser Gly Glu Asn Leu 
1               5                   10                  15      


Tyr Phe Gln Gly Gly Gly Ile Thr Cys Pro Pro Pro Met Ser Val Glu 
            20                  25                  30          


His Ala Asp Ile Trp Val Lys Ser Tyr Ser Leu Tyr Ser Arg Glu Arg 
        35                  40                  45              


Tyr Ile Cys Asn Ser Gly Phe Lys Arg Lys Ala Gly Thr Ser Ser Leu 
    50                  55                  60                  


Thr Glu Cys Val Leu Asn Lys Ala Thr Asn Val Ala His Trp Thr Thr 
65                  70                  75                  80  


Pro Ser Leu Lys Cys Ile Arg Asp Pro Ala Leu Val His Gln Arg Pro 
                85                  90                  95      


Ala Pro Pro Ser Gly Gly Ser Gly Gly Gly Gly Ser Gly Gly Gly Ser 
            100                 105                 110         


Gly Gly Gly Gly Ser Leu Gln Asn Trp Val Asn Val Ile Ser Asp Leu 
        115                 120                 125             


Lys Lys Ile Glu Asp Leu Ile Gln Ser Met His Ile Asp Ala Thr Leu 
    130                 135                 140                 


Tyr Thr Glu Ser Asp Val His Pro Ser Cys Lys Val Thr Ala Met Lys 
145                 150                 155                 160 


Cys Phe Leu Leu Glu Leu Gln Val Ile Ser Leu Glu Ser Gly Asp Ala 
                165                 170                 175     


Ser Ile His Asp Thr Val Glu Asn Leu Ile Ile Leu Ala Asn Asn Ser 
            180                 185                 190         


Leu Ser Ser Asn Gly Asn Val Thr Glu Ser Gly Cys Lys Glu Cys Glu 
        195                 200                 205             


Glu Leu Glu Glu Lys Asn Ile Lys Glu Phe Leu Gln Ser Phe Val His 
    210                 215                 220                 


Ile Val Gln Met Phe Ile Asn Thr Ser 
225                 230             


<210>  4
<211>  268
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Sequence identification of anti-4-1BB PF31

<400>  4

Asp Ile Val Met Thr Gln Ser Pro Pro Thr Leu Ser Leu Ser Pro Gly 
1               5                   10                  15      


Glu Arg Val Thr Leu Ser Cys Arg Ala Ser Gln Ser Ile Ser Asp Tyr 
            20                  25                  30          


Leu His Trp Tyr Gln Gln Lys Pro Gly Gln Ser Pro Arg Leu Leu Ile 
        35                  40                  45              


Lys Tyr Ala Ser Gln Ser Ile Ser Gly Ile Pro Ala Arg Phe Ser Gly 
    50                  55                  60                  


Ser Gly Ser Gly Thr Asp Phe Thr Leu Thr Ile Ser Ser Leu Glu Pro 
65                  70                  75                  80  


Glu Asp Phe Ala Val Tyr Tyr Cys Gln Asp Gly His Ser Phe Pro Pro 
                85                  90                  95      


Thr Phe Gly Gly Gly Thr Lys Val Glu Ile Lys Gly Gly Gly Gly Ser 
            100                 105                 110         


Gly Gly Gly Gly Ser Gly Gly Gly Gly Ser Gly Gly Gly Gly Ser Gln 
        115                 120                 125             


Val Gln Leu Val Gln Ser Gly Ala Glu Val Lys Lys Pro Gly Ala Ser 
    130                 135                 140                 


Val Lys Val Ser Cys Lys Ala Ser Gly Tyr Thr Phe Ser Ser Tyr Trp 
145                 150                 155                 160 


Met His Trp Val Arg Gln Ala Pro Gly Gln Arg Leu Glu Trp Met Gly 
                165                 170                 175     


Glu Ile Asn Pro Gly Asn Gly His Thr Asn Tyr Ser Gln Lys Phe Gln 
            180                 185                 190         


Gly Arg Val Thr Ile Thr Val Asp Lys Ser Ala Ser Thr Ala Tyr Met 
        195                 200                 205             


Glu Leu Ser Ser Leu Arg Ser Glu Asp Thr Ala Val Tyr Tyr Cys Ala 
    210                 215                 220                 


Arg Ser Phe Thr Thr Ala Arg Ala Phe Ala Tyr Trp Gly Gln Gly Thr 
225                 230                 235                 240 


Leu Val Thr Val Ser Ser Gly Gly Gly Gly Ser Gly Gly Gly Gly Ser 
                245                 250                 255     


Leu Pro Glu Thr Gly Gly His His His His His His 
            260                 265             


<210>  5
<211>  132
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Sequence identification of SYR-(G4S)3-IL15 (PF18)

<400>  5

Ser Tyr Arg Gly Gly Gly Gly Ser Gly Gly Gly Gly Ser Gly Gly Gly 
1               5                   10                  15      


Gly Ser Asn Trp Val Asn Val Ile Ser Asp Leu Lys Lys Ile Glu Asp 
            20                  25                  30          


Leu Ile Gln Ser Met His Ile Asp Ala Thr Leu Tyr Thr Glu Ser Asp 
        35                  40                  45              


Val His Pro Ser Cys Lys Val Thr Ala Met Lys Cys Phe Leu Leu Glu 
    50                  55                  60                  


Leu Gln Val Ile Ser Leu Glu Ser Gly Asp Ala Ser Ile His Asp Thr 
65                  70                  75                  80  


Val Glu Asn Leu Ile Ile Leu Ala Asn Asn Ser Leu Ser Ser Asn Gly 
                85                  90                  95      


Asn Val Thr Glu Ser Gly Cys Lys Glu Cys Glu Glu Leu Glu Glu Lys 
            100                 105                 110         


Asn Ile Lys Glu Phe Leu Gln Ser Phe Val His Ile Val Gln Met Phe 
        115                 120                 125             


Ile Asn Thr Ser 
    130         


<210>  6
<211>  229
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Sequence identification of SYR-(G4S)3-IL15R?-linker-IL15 (PF26)

<400>  6

Ser Tyr Arg Gly Gly Gly Gly Ser Gly Gly Gly Gly Ser Gly Gly Gly 
1               5                   10                  15      


Gly Ser Ile Thr Cys Pro Pro Pro Met Ser Val Glu His Ala Asp Ile 
            20                  25                  30          


Trp Val Lys Ser Tyr Ser Leu Tyr Ser Arg Glu Arg Tyr Ile Cys Asn 
        35                  40                  45              


Ser Gly Phe Lys Arg Lys Ala Gly Thr Ser Ser Leu Thr Glu Cys Val 
    50                  55                  60                  


Leu Asn Lys Ala Thr Asn Val Ala His Trp Thr Thr Pro Ser Leu Lys 
65                  70                  75                  80  


Cys Ile Arg Asp Pro Ala Leu Val His Gln Arg Pro Ala Pro Pro Ser 
                85                  90                  95      


Gly Gly Ser Gly Gly Gly Gly Ser Gly Gly Gly Ser Gly Gly Gly Gly 
            100                 105                 110         


Ser Leu Gln Asn Trp Val Asn Val Ile Ser Asp Leu Lys Lys Ile Glu 
        115                 120                 125             


Asp Leu Ile Gln Ser Met His Ile Asp Ala Thr Leu Tyr Thr Glu Ser 
    130                 135                 140                 


Asp Val His Pro Ser Cys Lys Val Thr Ala Met Lys Cys Phe Leu Leu 
145                 150                 155                 160 


Glu Leu Gln Val Ile Ser Leu Glu Ser Gly Asp Ala Ser Ile His Asp 
                165                 170                 175     


Thr Val Glu Asn Leu Ile Ile Leu Ala Asn Asn Ser Leu Ser Ser Asn 
            180                 185                 190         


Gly Asn Val Thr Glu Ser Gly Cys Lys Glu Cys Glu Glu Leu Glu Glu 
        195                 200                 205             


Lys Asn Ile Lys Glu Phe Leu Gln Ser Phe Val His Ile Val Gln Met 
    210                 215                 220                 


Phe Ile Asn Thr Ser 
225                 


