               SEQUENCE LISTING

<110> Ecole Polytechnique Federale de Lausanne (EPFL)
      Inserm Transfert SA

<120> Novel inhibitors of kallikrein proteases and uses thereof

<130> AC2196 PCT
 
<150> EP 19186320.8
<151> 2019-07-19

<160> 119

<170> BiSSAP 1.3

<210> 1
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7) 035

<400> 1
Gly Cys Thr Arg Gln Tyr Pro Cys 
1               5               

<210> 2
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7) 114

<400> 2
Pro Cys Leu Tyr Leu Ala Arg Cys 
1               5               

<210> 3
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3) 001

<400> 3
Gly Cys Thr Arg Gln Val Cys Gln Gln Thr Pro Ala Cys Pro Ser Ala 
1               5                   10                  15      
Cys Asn 
        

<210> 4
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3) 002

<400> 4
Gly Cys Thr Arg Gln Trp Pro Cys Asp Ser Val Pro Gly Ser Cys Thr 
1               5                   10                  15      
Cys Val 
        

<210> 5
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3) 003

<400> 5
Ala Cys Thr Arg Glu Tyr Asn Pro Gln Cys Ala Asn Pro Gln Cys Leu 
1               5                   10                  15      
Cys His 
        

<210> 6
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7) 004

<400> 6
Gly Cys Thr Arg Gln Trp Pro Cys Asp Ser Val Pro Gly Ser Cys Thr 
1               5                   10                  15      
Cys Val 
        

<210> 7
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7) 005

<400> 7
Ala Cys Thr Arg Glu Tyr Asn Pro Gln Cys Ala Asn Pro Gln Cys Leu 
1               5                   10                  15      
Cys His 
        

<210> 8
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7) 006

<400> 8
Met Cys Ser Arg Gln Trp Asp Pro Ser Leu Cys Cys Pro Gln Arg Thr 
1               5                   10                  15      
Cys Pro 
        

<210> 9
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7) 007

<400> 9
Arg Cys Asp Ser Ser Gln Cys Met Gln Gly Gln Cys Leu Tyr Arg Ser 
1               5                   10                  15      
Cys Pro 
        

<210> 10
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 008

<400> 10
His Cys Arg Lys Gly Leu Asp Arg Cys Pro Gln Cys Leu Tyr Arg Thr 
1               5                   10                  15      
Cys Ser 
        

<210> 11
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 009

<400> 11
Gln Cys Leu Tyr Ile Ala Cys Pro Ser Ala Ala Lys Cys Asp Asn Gly 
1               5                   10                  15      
Cys Gln 
        

<210> 12
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 010

<400> 12
Gln Cys Ile Ile Thr Tyr Gln Phe Cys Thr His Asp Arg Tyr Gly Cys 
1               5                   10                  15      
Cys Ser 
        

<210> 13
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7) 011

<400> 13
Arg Cys Phe Trp Gly Ala Arg Ser Thr Ser Gln Cys Asn Gln His Cys 
1               5                   10                  15      
Cys Glu 
        

<210> 14
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7) 012

<400> 14
Phe Cys Leu Trp Pro Trp Cys Gln Pro Pro Glu Ala Cys Pro Ser Gln 
1               5                   10                  15      
Cys Glu 
        

<210> 15
<211> 7
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3) 026

<400> 15
Gly Cys Thr Arg Gln Val Cys 
1               5           

<210> 16
<211> 7
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3) 027

<400> 16
Gly Cys Thr Arg Glu Val Cys 
1               5           

<210> 17
<211> 7
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3) 028

<400> 17
Gly Cys Thr Arg Gln Trp Cys 
1               5           

<210> 18
<211> 7
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3) 029

<400> 18
Gly Cys Thr Arg Glu Trp Cys 
1               5           

<210> 19
<211> 7
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3) 144

<400> 19
Gly Cys Ser Arg Gln Val Cys 
1               5           

<210> 20
<211> 9
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3) 031

<400> 20
Gly Cys Thr Arg Gln Trp Asp Pro Cys 
1               5                   

<210> 21
<211> 10
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3) 051

<400> 21
Gly Cys Thr Arg Gln Trp Asp Pro Ser Cys 
1               5                   10  

<210> 22
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7) 033

<400> 22
Gly Cys Thr Arg Gln Trp Pro Cys 
1               5               

<210> 23
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7) 034

<400> 23
Gly Cys Thr Arg Glu Trp Pro Cys 
1               5               

<210> 24
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7) 036

<400> 24
Gly Cys Thr Arg Glu Tyr Pro Cys 
1               5               

<210> 25
<211> 9
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7) 032

<400> 25
Gly Cys Thr Arg Gln Trp Pro Cys Asp 
1               5                   

<210> 26
<211> 9
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7) 039

<400> 26
Gly Cys Thr Arg Gln Trp Asp Pro Cys 
1               5                   

<210> 27
<211> 11
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7) 054

<400> 27
Gly Cys Thr Arg Gln Trp Asp Pro Ser Leu Cys 
1               5                   10      

<210> 28
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 080

<400> 28
Pro Cys Leu Tyr Leu Ser Cys Ser 
1               5               

<210> 29
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 081

<400> 29
Gln Cys Leu Tyr Leu Ser Cys Ser 
1               5               

<210> 30
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 082

<400> 30
Arg Cys Leu Tyr Leu Ser Cys Ser 
1               5               

<210> 31
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 083

<400> 31
Pro Cys Leu Phe Leu Ser Cys Ser 
1               5               

<210> 32
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 085

<400> 32
Pro Cys Leu Tyr Gln Ser Cys Ser 
1               5               

<210> 33
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 086

<400> 33
Pro Cys Leu Tyr Arg Ser Cys Ser 
1               5               

<210> 34
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 087

<400> 34
Pro Cys Leu Tyr Leu Ala Cys Ser 
1               5               

<210> 35
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 088

<400> 35
Pro Cys Leu Tyr Leu Thr Cys Ser 
1               5               

<210> 36
<211> 8
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 089

<400> 36
Pro Cys Leu Tyr Leu Ser Cys Pro 
1               5               

<210> 37
<211> 7
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 108

<400> 37
Cys Leu Tyr Leu Ala Cys Ser 
1               5           

<210> 38
<211> 7
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3) 109

<400> 38
Pro Cys Leu Tyr Leu Ala Cys 
1               5           

<210> 39
<211> 9
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7) 111

<400> 39
Pro Cys Leu Tyr Met Ala Arg Cys Ser 
1               5                   

<210> 40
<211> 9
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7) 112

<400> 40
Pro Cys Leu Tyr Leu Ala Gln Cys Ser 
1               5                   

<210> 41
<211> 9
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7) 095

<400> 41
Pro Cys Leu Tyr Leu Ser Arg Cys Ser 
1               5                   

<210> 42
<211> 9
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7) 096

<400> 42
Pro Cys Leu Tyr Leu Ala Arg Cys Ser 
1               5                   

<210> 43
<211> 7
<212> PRT
<213> Artificial Sequence

<220> 
<223> Heptapeptide linker

<400> 43
Glu Tyr Glu Lys Glu Tyr Glu 
1               5           

<210> 44
<211> 7
<212> PRT
<213> Artificial Sequence

<220> 
<223> Ser tag

<400> 44
Ser Ser Ser Lys Ser Ser Ser 
1               5           

<210> 45
<211> 7
<212> PRT
<213> Artificial Sequence

<220> 
<223> Flag epitope

<400> 45
Asp Tyr Lys Asp Asp Asp Lys 
1               5           

<210> 46
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 46
Gly Cys Ser Arg Gln Val Cys Gly Ile Cys Ser Pro Leu Ala Gln Ile 
1               5                   10                  15      
Cys Phe 
        

<210> 47
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 47
Gly Cys Thr Arg Glu Val Cys Trp Ser Ala Cys Ser Thr Gly Glu Gln 
1               5                   10                  15      
Cys Gln 
        

<210> 48
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 48
Gly Cys Ser Arg Glu Val Cys Tyr Ala Pro Ser Cys Gly Gln Ala Arg 
1               5                   10                  15      
Cys Gln 
        

<210> 49
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 49
Gly Cys Thr Arg Gln Ala Cys Ala Thr Val Gln Cys Leu Asn Tyr Gly 
1               5                   10                  15      
Cys Leu 
        

<210> 50
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 50
Ala Cys Thr Arg Gln Trp Cys Pro Glu Thr Pro Asn Cys Glu Pro Gly 
1               5                   10                  15      
Cys Leu 
        

<210> 51
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 51
Thr Cys Thr Arg Gln Trp Cys Gly Val Thr His His Cys Ala Asp Ser 
1               5                   10                  15      
Cys Asn 
        

<210> 52
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 52
Tyr Cys Thr Arg Gln Trp Cys Val Asn Leu Glu Asn Thr Cys Asp Thr 
1               5                   10                  15      
Cys Asp 
        

<210> 53
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 53
Glu Cys Thr Arg Gln Trp Cys Thr Val Thr Ala Ser Thr Ile Cys Ala 
1               5                   10                  15      
Cys Thr 
        

<210> 54
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 54
Phe Cys Thr Arg Glu Val Cys Ser Lys Gln Asp Ser Asn Thr Gln Cys 
1               5                   10                  15      
Cys Met 
        

<210> 55
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 55
Gly Cys Ser Arg Gln Ala Cys Ser Ser Trp Gln Leu Ile Gly Asn Cys 
1               5                   10                  15      
Cys Asp 
        

<210> 56
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 56
Gly Cys Thr Arg Gln Ala Thr Cys Ala Val Cys Gln Asp Asp Lys Ser 
1               5                   10                  15      
Cys Asn 
        

<210> 57
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 57
Ser Cys Thr Arg Glu Trp Trp Cys Pro Ser Ser Val Phe Val Ser Cys 
1               5                   10                  15      
Cys Gln 
        

<210> 58
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 58
Trp Cys Thr Arg Gln Tyr Pro Cys Asp Pro Pro Arg Pro Pro Thr Cys 
1               5                   10                  15      
Cys His 
        

<210> 59
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 59
Gly Cys Ser Arg Gln Trp Asp Gly Cys His Leu Asp Cys Pro Lys Gly 
1               5                   10                  15      
Cys Leu 
        

<210> 60
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 60
Gly Cys Thr Arg Gln Trp Thr Pro Cys Ala Gly Ser Tyr Cys Arg Asp 
1               5                   10                  15      
Cys Gln 
        

<210> 61
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 61
Gly Cys Thr Arg Glu Val Lys Gln Cys Pro Ala Gln Thr Cys Leu Thr 
1               5                   10                  15      
Cys Val 
        

<210> 62
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 62
Tyr Cys Ser Arg Glu Phe Asp Pro Ala Cys Gln Ser Leu Cys Ile Ser 
1               5                   10                  15      
Cys Phe 
        

<210> 63
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 63
Gly Cys Thr Arg Gln Tyr Gly Gly Gln Cys Cys Ser Gly Phe Trp Phe 
1               5                   10                  15      
Cys Glu 
        

<210> 64
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 3)

<400> 64
Gly Cys Thr Arg Glu Ala Asp Pro Thr Cys Leu Lys Met Cys Ala Gln 
1               5                   10                  15      
Cys Leu 
        

<210> 65
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 65
Ala Cys Thr Arg Gln Trp Pro Cys Trp Ser Glu Cys Leu Ser Leu Pro 
1               5                   10                  15      
Cys Ser 
        

<210> 66
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 66
Gly Cys Thr Arg Gln Tyr Pro Cys Met Thr Glu Pro Cys Leu Ala Ile 
1               5                   10                  15      
Cys Asp 
        

<210> 67
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 67
Arg Cys Thr Arg Glu Tyr Pro Cys Gln Pro Pro Met Pro Cys Gly Ser 
1               5                   10                  15      
Cys His 
        

<210> 68
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 68
Trp Cys Thr Arg Gln Tyr Pro Cys Asp Pro Pro Arg Pro Pro Thr Cys 
1               5                   10                  15      
Cys His 
        

<210> 69
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 69
Ser Cys Thr Arg Glu Trp Trp Cys Pro Ser Ser Val Phe Val Ser Cys 
1               5                   10                  15      
Cys Gln 
        

<210> 70
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 70
Phe Cys Thr Arg Glu Phe Leu Gly Cys Ser Pro Phe Cys Phe Val Gln 
1               5                   10                  15      
Cys Ala 
        

<210> 71
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 71
Ser Cys Thr Arg Glu Tyr Leu Gln Cys Pro Thr Phe Asp Asn Asp Cys 
1               5                   10                  15      
Cys Val 
        

<210> 72
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 72
Gly Cys Thr Arg Gln Tyr Gly Gly Gln Cys Cys Ser Gly Phe Trp Phe 
1               5                   10                  15      
Cys Glu 
        

<210> 73
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 73
Thr Cys Thr Arg Glu Trp Ala Gly Trp Cys Cys Thr Asn Glu Gln Pro 
1               5                   10                  15      
Cys Pro 
        

<210> 74
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 74
Gln Cys Thr Arg Glu Trp Leu Gly Thr Cys Ala Leu Cys Thr Thr Pro 
1               5                   10                  15      
Cys Tyr 
        

<210> 75
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 75
Gly Cys Thr Arg Gln Phe Pro Val Val Cys Met Pro Leu Cys Ser Val 
1               5                   10                  15      
Cys Thr 
        

<210> 76
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 76
Gly Cys Thr Arg Gln Phe Pro Gly Pro Trp Cys Gly Gly Ala Gly Cys 
1               5                   10                  15      
Cys Gln 
        

<210> 77
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 77
Ala Cys Thr Arg Asp Phe Asp Pro Trp His Cys Cys Ile Gln Arg Met 
1               5                   10                  15      
Cys Gln 
        

<210> 78
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 78
Gly Cys Thr Arg Asp Tyr Pro Leu Ser Asn Cys Gln Pro Cys Gln Lys 
1               5                   10                  15      
Cys Met 
        

<210> 79
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 79
Gly Cys Thr Arg Glu Trp Gln Tyr Pro Gly Cys Cys Tyr Ser Val Tyr 
1               5                   10                  15      
Cys Ile 
        

<210> 80
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 80
Gly Cys Thr Arg Gln Tyr Val Pro Gly Phe Ala Cys Ala Cys Gly Tyr 
1               5                   10                  15      
Cys Asp 
        

<210> 81
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 81
Thr Cys Thr Arg Glu Trp Phe Val Ser Gln Thr Cys Ile Cys Gln Ser 
1               5                   10                  15      
Cys His 
        

<210> 82
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 82
Gly Cys Thr Arg Asp Tyr Asp Phe Ser Ala Gln Cys Pro Gly Cys Arg 
1               5                   10                  15      
Cys Gly 
        

<210> 83
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK5 (Linker 7)

<400> 83
Gln Cys Thr Arg Gln Trp Asp Gly His Gly Val Cys Gly Pro Cys Gly 
1               5                   10                  15      
Cys Trp 
        

<210> 84
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 84
Arg Cys Gly Pro Thr Pro Cys Arg Ser Leu Pro Cys Leu Tyr Gln Ile 
1               5                   10                  15      
Cys Gln 
        

<210> 85
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 85
Ser Cys Ile Pro Pro Glu Cys Lys Ala Gly Val Cys Leu Tyr Gln Trp 
1               5                   10                  15      
Cys Arg 
        

<210> 86
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 86
Gln Cys Pro Ala Pro Ala Cys Ser Arg Val Pro Cys Leu Phe Ile Gly 
1               5                   10                  15      
Cys Gln 
        

<210> 87
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 87
Glu Cys Gln Ser Trp Pro Cys Asn Lys His Pro Cys Leu Tyr Leu Pro 
1               5                   10                  15      
Cys Pro 
        

<210> 88
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 88
Ala Cys Ala Glu Ser Thr Thr Cys Leu Gly Gln Cys Leu Tyr Arg Ser 
1               5                   10                  15      
Cys Gly 
        

<210> 89
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 89
Ala Cys Asp Pro Arg Gln Ser Cys Arg Ser Arg Cys Leu Tyr Gln His 
1               5                   10                  15      
Cys Ile 
        

<210> 90
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 90
Arg Cys Val Ala Tyr Arg Pro Cys Lys Pro Pro Cys Leu Tyr Ser Ser 
1               5                   10                  15      
Cys Ala 
        

<210> 91
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 91
Cys Cys Val Glu Ala Gly Arg Cys Ala Arg Gln Cys Leu Phe Leu Val 
1               5                   10                  15      
Cys Arg 
        

<210> 92
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 92
Ser Cys Ser Trp Ile Gly Arg Gln Cys Val Pro Cys Leu Phe Leu Ala 
1               5                   10                  15      
Cys Ser 
        

<210> 93
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 93
Lys Cys Gly Asn Gln Gly Asn Gln Cys Arg Arg Cys Leu Tyr Ser Ala 
1               5                   10                  15      
Cys Thr 
        

<210> 94
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 94
Ser Cys Arg Asp Gly Ser Gln Arg Cys Gly Arg Cys Leu Tyr Thr Ile 
1               5                   10                  15      
Cys Ser 
        

<210> 95
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 95
Arg Cys Leu Tyr Ile Thr Cys Cys Ser Gln Asp Gln Thr Thr Tyr Thr 
1               5                   10                  15      
Cys Gln 
        

<210> 96
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 96
Thr Cys Leu Ser His Thr Cys Pro Gln Cys Leu Tyr Leu His Asn Ser 
1               5                   10                  15      
Cys Ile 
        

<210> 97
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 97
Gln Cys Leu Tyr Ile Ala Cys Thr Pro Thr Glu His Cys Asn His Asp 
1               5                   10                  15      
Cys Arg 
        

<210> 98
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 98
Gln Cys Leu Tyr Ser Val Cys Ser Gly His Pro Gln Cys Pro Pro Thr 
1               5                   10                  15      
Cys Pro 
        

<210> 99
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 99
Gln Cys Leu Tyr Ala Val Cys His His Glu Ser Pro Cys Pro Ala Leu 
1               5                   10                  15      
Cys Ile 
        

<210> 100
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 3)

<400> 100
Gln Cys Leu Tyr Thr Ser Cys Asn Arg Trp Cys Pro Arg Ser Ala Thr 
1               5                   10                  15      
Cys Ala 
        

<210> 101
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 101
Gln Cys Leu Tyr Met Ala Arg Cys Ser Pro Val Cys Pro Gln Gln Tyr 
1               5                   10                  15      
Cys Gln 
        

<210> 102
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 102
Leu Cys Leu Tyr Leu Ala Gln Cys Gly Gly Arg Asp Lys Asp Cys Asp 
1               5                   10                  15      
Cys Val 
        

<210> 103
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 103
His Cys Leu Tyr Leu Gly His Ser Ser Cys Leu Cys Tyr Ser His Gln 
1               5                   10                  15      
Cys Ile 
        

<210> 104
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 104
Ile Cys Leu Tyr His Gly Arg Ser Glu Cys Cys His Tyr Ser Ala Gln 
1               5                   10                  15      
Cys Thr 
        

<210> 105
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 105
Leu Cys Leu Tyr Val Trp Pro Pro Ala Gly Ser Lys Cys Cys Gln Gln 
1               5                   10                  15      
Cys Gly 
        

<210> 106
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 106
Arg Cys Thr Ile Leu Tyr Ser Asn Cys Gln Ser Ala Pro Ser Arg Cys 
1               5                   10                  15      
Cys Ser 
        

<210> 107
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 107
Gln Cys Arg Thr Thr Tyr Gln Ala Cys Gly Ser Asn Ser Leu Gln Cys 
1               5                   10                  15      
Cys Asn 
        

<210> 108
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 108
Leu Cys Ile Thr Thr Tyr Gln Arg Thr Cys Pro Cys Ala Thr Pro Lys 
1               5                   10                  15      
Cys Arg 
        

<210> 109
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 109
Gln Cys Val Val Leu Tyr Gln Trp Pro Pro Cys Gln Cys Glu Thr Leu 
1               5                   10                  15      
Cys Val 
        

<210> 110
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 110
Trp Cys Val Thr Thr Tyr Met Asn Ala Ser Gly Cys Ser Asn Gln Cys 
1               5                   10                  15      
Cys Pro 
        

<210> 111
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 111
Leu Cys Val Gln Leu Tyr His Asn Asn Asp Ser Arg Cys Cys Ser Ser 
1               5                   10                  15      
Cys His 
        

<210> 112
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 112
Lys Cys Ile Ser Leu Tyr Leu Leu Pro Asn Pro Ser Cys Gln Ser Cys 
1               5                   10                  15      
Cys Thr 
        

<210> 113
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 113
Ser Cys Ile Ser Leu Tyr Gln Arg Val Gly Leu Ala Pro Cys Cys Trp 
1               5                   10                  15      
Cys Phe 
        

<210> 114
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 114
Ile Cys Phe Trp Gly Ala Arg Leu Cys Gln Pro Ala Cys Asn Pro Leu 
1               5                   10                  15      
Cys Ser 
        

<210> 115
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 115
Ser Cys Phe Trp Gly Ala Arg Thr Ser Cys Glu Pro Arg Gln Cys Pro 
1               5                   10                  15      
Cys Leu 
        

<210> 116
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 116
Arg Cys Phe Trp His Ala Arg Ser Thr Ser Pro Cys Thr His His Cys 
1               5                   10                  15      
Cys Ala 
        

<210> 117
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 117
Gln Cys Leu Trp Pro Trp Cys Cys Tyr Gln Ser Pro Asp His Gln Gly 
1               5                   10                  15      
Cys Ser 
        

<210> 118
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 118
Leu Cys Leu Trp Pro Trp Cys Gln Cys Ser Asn Pro Arg Pro Ser Asp 
1               5                   10                  15      
Cys His 
        

<210> 119
<211> 18
<212> PRT
<213> Artificial Sequence

<220> 
<223> KLK7 (Linker 7)

<400> 119
Leu Cys Leu Trp Pro Ala Cys Gly Pro Pro Pro Thr Cys Gly Ser Gln 
1               5                   10                  15      
Cys Thr 
        

