                         SEQUENCE LISTING

<110>  UNIVERSITY OF MARYLAND, BALTIMORE
 
<120>  SMALL MOLECULE INHIBITORS OF GPCR GPR68 AND RELATED RECEPTORS FOR
        TREATING CANCER, GLIOBLASTOMA, AND OTHER INDICATIONS

<130>  15024-364PC0

<140>  PCT/US2020/028651
<141>  2020-04-17

<150>  US 62/835,016
<151>  2019-04-17

<160>  16    

<170>  PatentIn version 3.5

<210>  1
<211>  16
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic: Rhodopsin


<220>
<221>  MOD_RES
<222>  (7)..(7)
<223>  PHOSPHORYLATION

<220>
<221>  MOD_RES
<222>  (9)..(9)
<223>  PHOSPHORYLATION

<400>  1

Gly Asp Asp Ala Ser Ala Thr Val Ser Lys Thr Glu Thr Ser Gln Val 
1               5                   10                  15      


<210>  2
<211>  17
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic: Vasopressin2


<220>
<221>  MOD_RES
<222>  (7)..(7)
<223>  PHOSPHORYLATION

<220>
<221>  MOD_RES
<222>  (9)..(9)
<223>  PHOSPHORYLATION

<220>
<221>  MOD_RES
<222>  (10)..(10)
<223>  PHOSPHORYLATION

<220>
<221>  MOD_RES
<222>  (13)..(13)
<223>  PHOSPHORYLATION

<400>  2

Ser Leu Gly Gln Asp Glu Ser Cys Thr Thr Ala Ser Ser Ser Leu Ala 
1               5                   10                  15      


Lys 
    


<210>  3
<211>  17
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic: GPR68


<220>
<221>  MOD_RES
<222>  (7)..(7)
<223>  PHOSPHORYLATION

<220>
<221>  MOD_RES
<222>  (10)..(10)
<223>  PHOSPHORYLATION

<400>  3

Pro Leu Gly Pro Glu Ala Ser Gly Lys Ser Gly Ala Gln Gly Glu Glu 
1               5                   10                  15      


Glu 
    


<210>  4
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic: rs1745752


<220>
<221>  misc_feature
<222>  (5)..(5)
<223>  Xaa can be any naturally occurring amino acid

<400>  4

Pro Leu Gly Pro Xaa 
1               5   


<210>  5
<211>  25
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: OGR1 morpholino

<400>  5
tttttccaac cacatgttca gagtc                                             25


<210>  6
<211>  25
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: Mismatch morpholino

<400>  6
cctcttacct cagttacaat ttata                                             25


<210>  7
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: GPR4 forward primer

<400>  7
ccctcctgtc ataattccat cc                                                22


<210>  8
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: GPR4 reverse primer

<400>  8
tggtctacag ggaagagatg ag                                                22


<210>  9
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: GPR65 forward primer

<400>  9
tggctgttgt ctaccctttg                                                   20


<210>  10
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: GPR65 reverse primer

<400>  10
ccacaacatg acagcattga ag                                                22


<210>  11
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: GPR68 forward primer

<400>  11
gtttgaaggc ggcagaaatg                                                   20


<210>  12
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: GPR68 reverse primer

<400>  12
gtggaatgag gaggcatgaa                                                   20


<210>  13
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: GPR132 forward primer

<400>  13
ttcaggagca tcaagcagag                                                   20


<210>  14
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: GPR132 reverse primer

<400>  14
cgaagcagac taggaagatg ac                                                22


<210>  15
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: GAPDH forward primer

<400>  15
gtttgaaggc ggcagaaatg                                                   20


<210>  16
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic: GAPDH reverse primer

<400>  16
gtggaatgag gaggcatgaa                                                   20


