                         SEQUENCE LISTING

<110>  Apros Therapeutics, Inc.
 
<120>  TLR7 PEPTIDE CONJUGATES

<130>  APTI-004/01WO 328217-2021

<150>  US 62/680,332
<151>  2018-06-04

<160>  24    

<170>  PatentIn version 3.5

<210>  1
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  1

His Ser Asn Leu Asn Asp Thr Thr Tyr Gln Arg Thr Arg Ala Leu Val 
1               5                   10                  15      


Arg Thr Gly Met Asp Pro Arg Met Cys 
            20                  25  


<210>  2
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  2

Lys Arg Lys Ser Ile Arg Ile Gln Arg Gly Pro Gly Arg Ala Phe Val 
1               5                   10                  15      


Thr Gly Lys Ile Gly Asn Met Arg Gln 
            20                  25  


<210>  3
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  3

Thr Leu Thr Cys Gly Phe Ala Asp Leu Met Gly Tyr Ile Pro Leu Val 
1               5                   10                  15      


Gly Ala Pro Leu Gly Gly Ala Ala Arg 
            20                  25  


<210>  4
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  4

Gly Leu Leu Leu Val Leu Ile Tyr Leu Tyr Gly Pro Ser Leu Tyr Arg 
1               5                   10                  15      


Arg Phe Phe Ser Asn Asp Cys Cys Ser 
            20                  25  


<210>  5
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  5

Asn Arg Phe Val Ser Ile Phe Ala Ser Gly Pro Ser Gln Lys Ile Gln 
1               5                   10                  15      


Leu Val Asn Asn Asn Gly Ser Trp His 
            20                  25  


<210>  6
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  6

Lys Arg Lys Ser Ile Arg Ile Gln Arg Gly Pro Gly Arg Ala Phe Val 
1               5                   10                  15      


Thr Ile Gly Lys Ile Gly Asn Met Arg 
            20                  25  


<210>  7
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  7

Asp Thr Ile Trp Ala Leu Ser Val Lys Tyr Gly Val Ser Val Gln Asp 
1               5                   10                  15      


Ile Met Ser Trp Asn Asn Leu Ser Ser 
            20                  25  


<210>  8
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  8

Leu Gly Arg Leu Met Tyr Asp Met Tyr Pro His Phe Met Pro Thr Asn 
1               5                   10                  15      


Leu Gly Pro Ser Glu Lys Arg Val Trp 
            20                  25  


<210>  9
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  9

Leu Leu Thr Arg Ile Leu Thr Ile Pro Gln Ser Leu Asp Ser Trp Trp 
1               5                   10                  15      


Thr Ser Leu Asn Phe Leu Gly Gly Ser 
            20                  25  


<210>  10
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  10

Glu Ser Leu Lys Ile Ser Gln Ala Val His Ala Ala His Ala Glu Ile 
1               5                   10                  15      


Asn Glu Ala Gly Arg Glu Val Val Gly 
            20                  25  


<210>  11
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  11

Glu Gln Leu Ser Ser Val Ser Ser Phe Glu Arg Phe Glu Ile Phe Pro 
1               5                   10                  15      


Lys Glu Ser Ser Trp Pro Asn His Asn 
            20                  25  


<210>  12
<211>  25
<212>  PRT
<213>  Mus musculus

<400>  12

His Pro Val Thr Ile Gly Glu Cys Pro Lys Tyr Val Arg Ser Ala Lys 
1               5                   10                  15      


Leu Arg Met Val Thr Gly Leu Arg Asn 
            20                  25  


<210>  13
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  13

His Ser Asn Leu Asn Asp Thr Thr Tyr Gln Arg Thr Arg Ala Leu Val 
1               5                   10                  15      


Arg Thr Gly Met Asp Pro Arg Met Cys 
            20                  25  


<210>  14
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  14

Lys Arg Lys Ser Ile Arg Ile Gln Arg Gly Pro Gly Arg Ala Phe Val 
1               5                   10                  15      


Thr Gly Lys Ile Gly Asn Met Arg Gln 
            20                  25  


<210>  15
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  15

Thr Leu Thr Cys Gly Phe Ala Asp Leu Met Gly Tyr Ile Pro Leu Val 
1               5                   10                  15      


Gly Ala Pro Leu Gly Gly Ala Ala Arg 
            20                  25  


<210>  16
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  16

Gly Leu Leu Leu Val Leu Ile Tyr Leu Tyr Gly Pro Ser Leu Tyr Arg 
1               5                   10                  15      


Arg Phe Phe Ser Asn Asp Cys Cys Ser 
            20                  25  


<210>  17
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  17

Asn Arg Phe Val Ser Ile Phe Ala Ser Gly Pro Ser Gln Lys Ile Gln 
1               5                   10                  15      


Leu Val Asn Asn Asn Gly Ser Trp His 
            20                  25  


<210>  18
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  18

Lys Arg Lys Ser Ile Arg Ile Gln Arg Gly Pro Gly Arg Ala Phe Val 
1               5                   10                  15      


Thr Ile Gly Lys Ile Gly Asn Met Arg 
            20                  25  


<210>  19
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  19

Asp Thr Ile Trp Ala Leu Ser Val Lys Tyr Gly Val Ser Val Gln Asp 
1               5                   10                  15      


Ile Met Ser Trp Asn Asn Leu Ser Ser 
            20                  25  


<210>  20
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  20

Leu Gly Arg Leu Met Tyr Asp Met Tyr Pro His Phe Met Pro Thr Asn 
1               5                   10                  15      


Leu Gly Pro Ser Glu Lys Arg Val Trp 
            20                  25  


<210>  21
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  21

Leu Leu Thr Arg Ile Leu Thr Ile Pro Gln Ser Leu Asp Ser Trp Trp 
1               5                   10                  15      


Thr Ser Leu Asn Phe Leu Gly Gly Ser 
            20                  25  


<210>  22
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  22

Glu Ser Leu Lys Ile Ser Gln Ala Val His Ala Ala His Ala Glu Ile 
1               5                   10                  15      


Asn Glu Ala Gly Arg Glu Val Val Gly 
            20                  25  


<210>  23
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  23

Glu Gln Leu Ser Ser Val Ser Ser Phe Glu Arg Phe Glu Ile Phe Pro 
1               5                   10                  15      


Lys Glu Ser Ser Trp Pro Asn His Asn 
            20                  25  


<210>  24
<211>  25
<212>  PRT
<213>  Mus musculus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  conjugated to TLR7 agonist Compound 1

<400>  24

His Pro Val Thr Ile Gly Glu Cys Pro Lys Tyr Val Arg Ser Ala Lys 
1               5                   10                  15      


Leu Arg Met Val Thr Gly Leu Arg Asn 
            20                  25  


