                         SEQUENCE LISTING

<110>  INTENDET SERVICES, INC.
       GIROIR, Brett P.
       KERN, Clifford  H. III
       LEUSCHNER, Carola
 
<120>  IMMUNE-STIMULATING PEPTIDES AND CHECKPOINT INHIBITORS, AND USES THEREOF FOR TREATING CANCER

<130>  038524-0501516

<140>  PCT/US2018/063848
<141>  2018-12-04

<150>  62/594829
<151>  2017-12-05

<160>  45    

<170>  PatentIn version 3.5

<210>  1
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  1

Tyr Gly Gly Phe 
1               


<210>  2
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  2

Tyr Gly Gly Trp 
1               


<210>  3
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  3

Tyr Gly Gly Phe Gly Gly Phe Gly 
1               5               


<210>  4
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (7)..(7)
<223>  Xaa is Dip (3,3-diphenylalanine)

<400>  4

Tyr Gly Gly Phe Gly Gly Xaa Gly 
1               5               


<210>  5
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (7)..(7)
<223>  Xaa is Bip (biphenylalanine)

<400>  5

Tyr Gly Gly Phe Gly Gly Xaa Gly 
1               5               


<210>  6
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (7)..(7)
<223>  Xaa is Ath (9-anthracenylalanine)

<400>  6

Tyr Gly Gly Phe Gly Gly Xaa Gly 
1               5               


<210>  7
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (7)..(7)
<223>  Xaa is Dap (2,3-diaminopropionic acid)

<400>  7

Tyr Gly Gly Phe Gly Gly Xaa Gly 
1               5               


<210>  8
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (7)..(7)
<223>  Xaa is Dab (2,4-diaminobutanoic acid)

<400>  8

Tyr Gly Gly Phe Gly Gly Xaa Gly 
1               5               


<210>  9
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (7)..(7)
<223>  Xaa is Nal (1- naphthylalanine)

<400>  9

Tyr Gly Gly Phe Gly Gly Xaa Gly 
1               5               


<210>  10
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  10

Tyr Gly Gly Trp Gly Gly Phe Gly 
1               5               


<210>  11
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  11

Tyr Gly Gly Trp Gly Gly Trp Gly 
1               5               


<210>  12
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  12

Tyr Gly Gly Phe Met 
1               5   


<210>  13
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Dip (3,3-diphenylalanine)

<400>  13

Tyr Gly Gly Xaa Met 
1               5   


<210>  14
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Bip (biphenylalanine)

<400>  14

Tyr Gly Gly Xaa Met 
1               5   


<210>  15
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Ath (9-anthracenylalanine)

<400>  15

Tyr Gly Gly Xaa Met 
1               5   


<210>  16
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Dap (2,3-diaminopropionic acid)

<400>  16

Tyr Gly Gly Xaa Met 
1               5   


<210>  17
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Dab (2,4-diaminobutanoic acid)

<400>  17

Tyr Gly Gly Xaa Met 
1               5   


<210>  18
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Nal (1- naphthylalanine)

<400>  18

Tyr Gly Gly Xaa Met 
1               5   


<210>  19
<211>  9
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  19

Tyr Gly Gly Trp Met Tyr Gly Ala Phe 
1               5                   


<210>  20
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  20

Tyr Gly Ala Trp 
1               


<210>  21
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (3)..(3)
<223>  Xaa is Aib (Alpha-aminoisobutyric acid)

<400>  21

Tyr Gly Xaa Phe Met 
1               5   


<210>  22
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Dip (3,3-diphenylalanine)

<400>  22

Tyr Gly Ala Xaa Met 
1               5   


<210>  23
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Bip (biphenylalanine)

<400>  23

Tyr Gly Ala Xaa Met 
1               5   


<210>  24
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Ath (9-anthracenylalanine)

<400>  24

Tyr Gly Ala Xaa Met 
1               5   


<210>  25
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Dap (2,3-diaminopropionic acid)

<400>  25

Tyr Gly Ala Xaa Met 
1               5   


<210>  26
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Dab (2,4-diaminobutanoic acid)

<400>  26

Tyr Gly Ala Xaa Met 
1               5   


<210>  27
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (4)..(4)
<223>  Xaa is Nal (1- naphthylalanine)

<400>  27

Tyr Gly Ala Xaa Met 
1               5   


<210>  28
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  28

Tyr Gly Gly Trp Met 
1               5   


<210>  29
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  29

Tyr Gly Ala Phe 
1               


<210>  30
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  30

Tyr Ala Gly Phe 
1               


<210>  31
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  31

Tyr Ala Gly Trp 
1               


<210>  32
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (2)..(2)
<223>  Xaa is Aib (Alpha-aminoisobutyric acid)

<400>  32

Tyr Xaa Gly Phe Met 
1               5   


<210>  33
<211>  9
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  33

Ala Cys Tyr Gly Gly Gly Ala Cys Gly 
1               5                   


<210>  34
<211>  9
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  34

Ala Cys Tyr Gly Gly Phe Ala Cys Gly 
1               5                   


<210>  35
<211>  9
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (6)..(6)
<223>  Xaa is Bip (biphenylalanine)

<400>  35

Ala Cys Tyr Gly Gly Xaa Ala Cys Gly 
1               5                   


<210>  36
<211>  9
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (6)..(6)
<223>  Xaa is Dip (3,3-diphenylalanine)

<400>  36

Ala Cys Tyr Gly Gly Xaa Ala Cys Gly 
1               5                   


<210>  37
<211>  9
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (6)..(6)
<223>  Xaa is Ath (9-anthracenylalanine)

<400>  37

Ala Cys Tyr Gly Gly Xaa Ala Cys Gly 
1               5                   


<210>  38
<211>  9
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (6)..(6)
<223>  Xaa is Dab (2,4-diaminobutanoic acid)

<400>  38

Ala Cys Tyr Gly Gly Xaa Ala Cys Gly 
1               5                   


<210>  39
<211>  9
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (6)..(6)
<223>  Xaa is Dap (2,3-diaminopropionic acid)

<400>  39

Ala Cys Tyr Gly Gly Xaa Ala Cys Gly 
1               5                   


<210>  40
<211>  9
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide


<220>
<221>  SITE
<222>  (6)..(6)
<223>  Xaa is Nal (1- naphthylalanine)

<400>  40

Ala Cys Tyr Gly Gly Xaa Ala Cys Gly 
1               5                   


<210>  41
<211>  9
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  41

Ala Cys Tyr Gly Gly Gly Trp Cys Gly 
1               5                   


<210>  42
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  42

Tyr Gly Gly Phe Leu 
1               5   


<210>  43
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  43

Tyr Gly Tyr Gly 
1               


<210>  44
<211>  6
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  44

Tyr Gly Tyr Gly Tyr Gly 
1               5       


<210>  45
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic immune-stimulating peptide

<400>  45

Tyr Gly Tyr Gly Tyr Gly Tyr Gly 
1               5               


