                         SEQUENCE LISTING

<110>  Fondation The Ark
 
<120>  FUSION RESPIRATORY SYNCYTIAL VIRUS INHIBITORS AND USE THEREOF

<130>  P1996PC00

<150>  16158364.6
<151>  2016-03-03

<160>  50    

<170>  PatentIn version 3.3

<210>  1
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Consensus


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  Any amino acid

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  selected from any amino acid or a cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (3)..(3)
<223>  apolar amino-acid

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  selected from any amino acid or a cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  selected from any amino acid or a cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (6)..(6)
<223>  Any amino acid

<220>
<221>  MISC_FEATURE
<222>  (7)..(7)
<223>  apolar amino-acid

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (9)..(9)
<223>  apolar amino-acid

<220>
<221>  MISC_FEATURE
<222>  (10)..(10)
<223>  apolar amino-acid

<220>
<221>  MISC_FEATURE
<222>  (11)..(12)
<223>  independently selected from a polar amino acid and a cross-linked
       amino-acid

<220>
<221>  MISC_FEATURE
<222>  (13)..(13)
<223>  Serine

<220>
<221>  MISC_FEATURE
<222>  (14)..(14)
<223>  Any amino acid

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  selected from a polar amino acid and a cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  apolar amino-acid

<220>
<221>  MISC_FEATURE
<222>  (17)..(17)
<223>  apolar amino-acid

<220>
<221>  MISC_FEATURE
<222>  (18)..(18)
<223>  Any amino acid

<220>
<221>  MISC_FEATURE
<222>  (19)..(19)
<223>  selected from any amino acid or a cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  apolar amino-acid

<400>  1

Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa 
1               5                   10                  15      


Xaa Xaa Xaa Xaa 
            20  


<210>  2
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  Consensus for 4bb


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (3)..(3)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (6)..(6)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (7)..(7)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  cross linked amino acid

<220>
<221>  MISC_FEATURE
<222>  (9)..(9)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (10)..(10)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  polar amino acid

<220>
<221>  MISC_FEATURE
<222>  (13)..(13)
<223>  Serine

<220>
<221>  MISC_FEATURE
<222>  (14)..(14)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (17)..(17)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (18)..(18)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (19)..(19)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  apolar amino acid

<400>  2

Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa 
1               5                   10                  15      


Xaa Xaa Xaa Xaa 
            20  


<210>  3
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  4bb spe


<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  cross-linked amino-acid

<400>  3

Glu Lys Ile Xaa Gln Ser Leu Xaa Phe Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  4
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4bb497


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  4

Ala Lys Ile Xaa Gln Ser Leu Xaa Phe Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  5
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>   V4bb498


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  5

Glu Ala Ile Xaa Gln Ser Leu Xaa Phe Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  6
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4bb499


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  6

Glu Lys Ala Xaa Gln Ser Leu Xaa Phe Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  7
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4a500


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (19)..(19)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  7

Glu Lys Ile Ala Gln Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Xaa Val 
            20  


<210>  8
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4bb501


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  8

Glu Lys Ile Xaa Ala Ser Leu Xaa Phe Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  9
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4bb502


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  9

Glu Lys Ile Xaa Gln Ala Leu Xaa Phe Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  10
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4bb503


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  10

Glu Lys Ile Xaa Gln Ser Ala Xaa Phe Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  11
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4bb505


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  11

Glu Lys Ile Xaa Gln Ser Leu Xaa Ala Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  12
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4bb510


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  12

Glu Lys Ile Xaa Gln Ser Leu Xaa Phe Ile Xaa Lys Ser Ala Xaa Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  13
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4bb512


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  13

Glu Lys Ile Xaa Gln Ser Leu Xaa Phe Ile Xaa Lys Ser Asp Xaa Ala 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  14
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4bb514


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  14

Glu Lys Ile Xaa Gln Ser Leu Xaa Phe Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu Ala Asn Val 
            20  


<210>  15
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4bb515


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  15

Glu Lys Ile Xaa Gln Ser Leu Xaa Phe Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Ala Val 
            20  


<210>  16
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4bb516


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  16

Glu Lys Ile Xaa Gln Ser Leu Xaa Phe Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Asn Ala 
            20  


<210>  17
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  Consensus for 4ca


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (3)..(3)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (6)..(6)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (7)..(7)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (9)..(9)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (10)..(10)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  polar amino acid

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (13)..(13)
<223>  Serine

<220>
<221>  MISC_FEATURE
<222>  (14)..(14)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  polar amino acid

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (17)..(17)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (18)..(18)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (19)..(19)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  apolar amino acid

<400>  17

Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa 
1               5                   10                  15      


Xaa Xaa Xaa Xaa 
            20  


<210>  18
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  4ca specific varied on staples


<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  cross-linked amino-acid

<400>  18

Glu Xaa Ile Asn Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  19
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  Peptide 4a


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (19)..(19)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  19

Glu Lys Ile Asn Gln Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Xaa Val 
            20  


<210>  20
<211>  17
<212>  PRT
<213>  Artificial sequence

<220>
<223>  Peptide 3ac


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (9)..(9)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (17)..(17)
<223>  C-term amidated

<400>  20

Glu Gln Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Xaa Leu Leu His Xaa 
1               5                   10                  15      


Val 
    


<210>  21
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  comparative peptide 4bf


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (R)-2-(7-octenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (19)..(19)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  21

Glu Lys Ile Xaa Gln Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Leu 
1               5                   10                  15      


Leu His Xaa Val 
            20  


<210>  22
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  Comparative peptide 4

<400>  22

Glu Lys Ile Asn Gln Ser Leu Ala Phe Ile Arg Lys Ser Asp Glu Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  23
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  Comparative peptide 4e


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (R)-2-(7-octenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  23

Glu Lys Ile Asn Gln Ser Leu Xaa Phe Ile Arg Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  24
<211>  49
<212>  PRT
<213>  Artificial sequence

<220>
<223>  HR2- fragment 476-524

<400>  24

Asn Phe Tyr Asp Pro Leu Val Phe Pro Ser Asp Glu Phe Asp Ala Ser 
1               5                   10                  15      


Ile Ser Gln Val Asn Glu Lys Ile Asn Gln Ser Leu Ala Phe Ile Arg 
            20                  25                  30          


Lys Ser Asp Glu Leu Leu His Asn Val Asn Ala Gly Lys Ser Thr Thr 
        35                  40                  45              


Asn 
    


<210>  25
<211>  38
<212>  PRT
<213>  Artificial sequence

<220>
<223>  X-ray of fragment 480-516

<400>  25

Pro Leu Val Phe Pro Ser Asp Glu Phe Asp Ala Ser Ile Ser Gln Val 
1               5                   10                  15      


Asn Glu Lys Ile Asn Gln Ser Leu Ala Phe Ile Arg Lys Ser Asp Glu 
            20                  25                  30          


Leu Leu His Asn Val Asn 
        35              


<210>  26
<211>  35
<212>  PRT
<213>  Artificial sequence

<220>
<223>  T108 fragment 478-512

<400>  26

Tyr Asp Pro Leu Val Phe Pro Ser Asp Glu Phe Asp Ala Ser Ile Ser 
1               5                   10                  15      


Gln Val Asn Glu Lys Ile Asn Gln Ser Leu Ala Phe Ile Arg Lys Ser 
            20                  25                  30          


Asp Glu Leu 
        35  


<210>  27
<211>  35
<212>  PRT
<213>  Artificial sequence

<220>
<223>  T118 fragment 488-522

<400>  27

Phe Asp Ala Ser Ile Ser Gln Val Asn Glu Lys Ile Asn Gln Ser Leu 
1               5                   10                  15      


Ala Phe Ile Arg Lys Ser Asp Glu Leu Leu His Asn Val Asn Ala Gly 
            20                  25                  30          


Lys Ser Thr 
        35  


<210>  28
<211>  35
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  SAFH-RSVFBD


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (3)..(3)
<223>  (R)-2-(7-octenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (10)..(10)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  (R)-2-(7-octenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (27)..(27)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (35)..(35)
<223>  C-term amidated

<400>  28

Phe Asp Xaa Ser Ile Ser Gln Val Asn Xaa Lys Ile Asn Gln Ser Leu 
1               5                   10                  15      


Ala Phe Ile Xaa Lys Ser Asp Glu Leu Leu Xaa Asn Val Asn Ala Gly 
            20                  25                  30          


Lys Ser Thr 
        35  


<210>  29
<211>  19
<212>  PRT
<213>  Artificial sequence

<220>
<223>  comparative peptide 1eg


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (9)..(9)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (19)..(19)
<223>  C-term amidated

<400>  29

Glu Phe Pro Ser Xaa Glu Phe Asp Xaa Ser Ile Xaa Gln Val Asn Xaa 
1               5                   10                  15      


Lys Ile Asn 
            


<210>  30
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  comparative peptide 4ef


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  (R)-2-(7-octenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (R)-2-(7-octenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (19)..(19)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  30

Xaa Lys Ile Asn Gln Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Leu 
1               5                   10                  15      


Leu His Xaa Val 
            20  


<210>  31
<211>  17
<212>  PRT
<213>  Artificial sequence

<220>
<223>  comparative peptide 3

<400>  31

Glu Gln Ser Leu Ala Phe Ile Arg Lys Ser Asp Glu Leu Leu His Asn 
1               5                   10                  15      


Val 
    


<210>  32
<211>  17
<212>  PRT
<213>  Artificial sequence

<220>
<223>  comparative peptide 3a


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (9)..(9)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (17)..(17)
<223>  C-term amidated

<400>  32

Glu Gln Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Leu Leu His Asn 
1               5                   10                  15      


Val 
    


<210>  33
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  Consensus for 4a


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  Any amino acid

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (3)..(3)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (3)..(3)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (6)..(6)
<223>  any amino acid

<220>
<221>  MISC_FEATURE
<222>  (7)..(7)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  cross-linked amino acid

<220>
<221>  MISC_FEATURE
<222>  (9)..(9)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (10)..(10)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  polar amino acid

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  cross-linked amino acid

<220>
<221>  MISC_FEATURE
<222>  (13)..(13)
<223>  Serine

<220>
<221>  MISC_FEATURE
<222>  (14)..(14)
<223>  Any amino acid

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  Cross-linked amino acid

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (17)..(17)
<223>  apolar amino acid

<220>
<221>  MISC_FEATURE
<222>  (18)..(18)
<223>  Any amino acid

<220>
<221>  MISC_FEATURE
<222>  (19)..(19)
<223>  Cross-linked amino acid

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  apolar amino acid

<400>  33

Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa Xaa 
1               5                   10                  15      


Xaa Xaa Xaa Xaa 
            20  


<210>  34
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  4a spe


<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  cross-linked amino-acid

<220>
<221>  MISC_FEATURE
<222>  (19)..(19)
<223>  cross-linked amino-acid

<400>  34

Glu Lys Ile Asn Gln Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Xaa Val 
            20  


<210>  35
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  4bb-4bb'


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine or (S)-2-(4-pentenyl)glycine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine or (S)-2-(4-pentenyl)glycine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine or (S)-2-(4-pentenyl)glycine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)alanine or (S)-2-(4-pentenyl)glycine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  35

Glu Lys Ile Xaa Gln Ser Leu Xaa Phe Ile Xaa Lys Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  36
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  36

Glu Xaa Ile Asn Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  37
<211>  20
<212>  PRT
<213>  Artificial sequence

<220>
<223>  V4ca511


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  37

Glu Xaa Ile Asn Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Ala Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  38
<211>  18
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca18


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (18)..(18)
<223>  C-term amidated

<400>  38

Glu Xaa Ile Asn Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Leu 
1               5                   10                  15      


Leu His 
        


<210>  39
<211>  16
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca16


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (7)..(7)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (11)..(11)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  C-term amidated

<400>  39

Xaa Ile Asn Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Leu Leu 
1               5                   10                  15      


<210>  40
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca-var1


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (7)..(7)
<223>  tBa

<220>
<221>  MISC_FEATURE
<222>  (7)..(7)
<223>  L-3-tButyl-Alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  40

Glu Xaa Ile Asn Xaa Ser Xaa Xaa Phe Ile Arg Xaa Ser Asp Glu Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  41
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca-var2


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (7)..(7)
<223>  L-2-Cyclopentyl-Glycine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  41

Glu Xaa Ile Asn Xaa Ser Xaa Xaa Phe Ile Arg Xaa Ser Asp Glu Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  42
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca-var3


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (7)..(7)
<223>  2-Cyclohexyl-L-Glycine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  42

Glu Xaa Ile Asn Xaa Ser Xaa Xaa Phe Ile Arg Xaa Ser Asp Glu Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  43
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca-var4


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  L-3-tButyl-Alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  43

Glu Xaa Ile Asn Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Xaa 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  44
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca-var5


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  L-3-tButyl-Alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  44

Glu Xaa Ile Lys Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Xaa 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  45
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca-var6


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  L-3-tButyl-Alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  45

Glu Xaa Ile Arg Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Xaa 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  46
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca-var7


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  3-Cyclohexyl-L-Alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  46

Glu Xaa Ile Asn Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Xaa 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  47
<211>  18
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca-var8


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  L-3-tButyl-Alanine

<220>
<221>  MISC_FEATURE
<222>  (18)..(18)
<223>  C-term amidated

<400>  47

Glu Xaa Ile Asn Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Xaa 
1               5                   10                  15      


Leu His 
        


<210>  48
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca-var9


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  L-3-tButyl-Alanine

<220>
<221>  MISC_FEATURE
<222>  (17)..(17)
<223>  L-3-tButyl-Alanine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  48

Glu Xaa Ile Asn Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Xaa 
1               5                   10                  15      


Xaa His Asn Val 
            20  


<210>  49
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4ca2


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  (R)-2-(4-pentenyl)alanine

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  (S)-2-(4-pentenyl)glycine

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)glycine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)glycine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  49

Glu Xaa Ile Asn Xaa Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Glu Leu 
1               5                   10                  15      


Leu His Asn Val 
            20  


<210>  50
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  4a2


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  N-term acetylated

<220>
<221>  MISC_FEATURE
<222>  (8)..(8)
<223>  (S)-2-(4-pentenyl)glycine

<220>
<221>  MISC_FEATURE
<222>  (12)..(12)
<223>  (S)-2-(4-pentenyl)glycine

<220>
<221>  MISC_FEATURE
<222>  (15)..(15)
<223>  (S)-2-(4-pentenyl)glycine

<220>
<221>  MISC_FEATURE
<222>  (19)..(19)
<223>  (S)-2-(4-pentenyl)glycine

<220>
<221>  MISC_FEATURE
<222>  (20)..(20)
<223>  C-term amidated

<400>  50

Glu Lys Ile Asn Gln Ser Leu Xaa Phe Ile Arg Xaa Ser Asp Xaa Leu 
1               5                   10                  15      


Leu His Xaa Val 
            20  


