                         SEQUENCE LISTING

<110>  New York University
       Arora, Paramjit S.
       Lao, Brooke Bullock
       Bonneau, Richard
       Drew, Kevin
 
<120>  OXOPIPERAZINE HELIX MIMETICS FOR CONTROL OF HYPOXIA-INDUCIBLE 
       GENE EXPRESSION

<130>  29527.1621 (ARO01-25PCT)

<140>  PCT/US2015/031816
<141>  2015-05-20

<150>  US 62/001,530
<151>  2014-05-21

<160>  5     

<170>  PatentIn version 3.5

<210>  1
<211>  51
<212>  PRT
<213>  Artificial

<220>
<223>  Human HIF1alpha C-terminal transactivation domain

<400>  1

Ser Asp Leu Ala Cys Arg Leu Leu Gly Gln Ser Met Asp Glu Ser Gly 
1               5                   10                  15      


Leu Pro Gln Leu Thr Ser Tyr Asp Cys Glu Val Asn Ala Pro Ile Gln 
            20                  25                  30          


Gly Ser Arg Asn Leu Leu Gln Gly Glu Glu Leu Leu Arg Ala Leu Asp 
        35                  40                  45              


Gln Val Asn 
    50      


<210>  2
<211>  29
<212>  PRT
<213>  Artificial

<220>
<223>  Signal peptide

<400>  2

Met Met Ser Phe Val Ser Leu Leu Leu Val Gly Ile Leu Phe Tyr Ala 
1               5                   10                  15      


Thr Glu Ala Glu Gln Leu Thr Lys Cys Glu Val Phe Gln 
            20                  25                  


<210>  3
<211>  4
<212>  PRT
<213>  Artificial

<220>
<223>  ER retention signal

<400>  3

Lys Glu Asp Leu 
1               


<210>  4
<211>  8
<212>  PRT
<213>  Artificial

<220>
<223>  Nuclear transport peptide

<400>  4

Pro Pro Lys Lys Lys Arg Lys Val 
1               5               


<210>  5
<211>  25
<212>  PRT
<213>  Artificial

<220>
<223>  Transport peptide

<400>  5

Met Leu Ser Leu Arg Gln Ser Ile Arg Phe Phe Lys Pro Ala Thr Arg 
1               5                   10                  15      


Thr Leu Cys Ser Ser Arg Tyr Leu Leu 
            20                  25  


