                               SEQUENCE LISTING

<110> MERRIMACK PHARMACEUTICALS, INC.
 
<120> DOSAGE AND ADMINISTRATION OF ANTI-EGFR THERAPEUTICS

<130> MMJ-046PC

<140>
<141>

<150> 62/005,401
<151> 2014-05-30

<150> 61/996,819
<151> 2014-05-14

<160> 24    

<170> PatentIn version 3.5

<210> 1
<211> 140
<212> PRT
<213> Homo sapiens

<400> 1
Met Gly Phe Gly Leu Ser Trp Leu Phe Leu Val Ala Ile Leu Lys Gly 
1               5                   10                  15      


Val Gln Cys Gln Val Gln Leu Val Gln Ser Gly Ala Glu Val Lys Lys 
            20                  25                  30          


Pro Gly Ser Ser Val Lys Val Ser Cys Lys Ala Ser Gly Gly Thr Phe 
        35                  40                  45              


Ser Ser Tyr Ala Ile Ser Trp Val Arg Gln Ala Pro Gly Gln Gly Leu 
    50                  55                  60                  


Glu Trp Met Gly Ser Ile Ile Pro Ile Phe Gly Thr Val Asn Tyr Ala 
65                  70                  75                  80  


Gln Lys Phe Gln Gly Arg Val Thr Ile Thr Ala Asp Glu Ser Thr Ser 
                85                  90                  95      


Thr Ala Tyr Met Glu Leu Ser Ser Leu Arg Ser Glu Asp Thr Ala Val 
            100                 105                 110         


Tyr Tyr Cys Ala Arg Asp Pro Ser Val Asn Leu Tyr Trp Tyr Phe Asp 
        115                 120                 125             


Leu Trp Gly Arg Gly Thr Leu Val Thr Val Ser Ser 
    130                 135                 140 


<210> 2
<211> 127
<212> PRT
<213> Homo sapiens

<400> 2
Met Gly Thr Pro Ala Gln Leu Leu Phe Leu Leu Leu Leu Trp Leu Pro 
1               5                   10                  15      


Asp Thr Thr Gly Asp Ile Gln Met Thr Gln Ser Pro Ser Thr Leu Ser 
            20                  25                  30          


Ala Ser Val Gly Asp Arg Val Thr Ile Thr Cys Arg Ala Ser Gln Ser 
        35                  40                  45              


Ile Ser Ser Trp Trp Ala Trp Tyr Gln Gln Lys Pro Gly Lys Ala Pro 
    50                  55                  60                  


Lys Leu Leu Ile Tyr Asp Ala Ser Ser Leu Glu Ser Gly Val Pro Ser 
65                  70                  75                  80  


Arg Phe Ser Gly Ser Gly Ser Gly Thr Glu Phe Thr Leu Thr Ile Ser 
                85                  90                  95      


Ser Leu Gln Pro Asp Asp Phe Ala Thr Tyr Tyr Cys Gln Gln Tyr His 
            100                 105                 110         


Ala His Pro Thr Thr Phe Gly Gly Gly Thr Lys Val Glu Ile Lys 
        115                 120                 125         


<210> 3
<211> 138
<212> PRT
<213> Homo sapiens

<400> 3
Met Gly Phe Gly Leu Ser Trp Leu Phe Leu Val Ala Ile Leu Lys Gly 
1               5                   10                  15      


Val Gln Cys Gln Val Gln Leu Val Gln Ser Gly Ala Glu Val Lys Lys 
            20                  25                  30          


Pro Gly Ser Ser Val Lys Val Ser Cys Lys Ala Ser Gly Gly Thr Phe 
        35                  40                  45              


Gly Ser Tyr Ala Ile Ser Trp Val Arg Gln Ala Pro Gly Gln Gly Leu 
    50                  55                  60                  


Glu Trp Met Gly Ser Ile Ile Pro Ile Phe Gly Ala Ala Asn Pro Ala 
65                  70                  75                  80  


Gln Lys Ser Gln Gly Arg Val Thr Ile Thr Ala Asp Glu Ser Thr Ser 
                85                  90                  95      


Thr Ala Tyr Met Glu Leu Ser Ser Leu Arg Ser Glu Asp Thr Ala Val 
            100                 105                 110         


Tyr Tyr Cys Ala Lys Met Gly Arg Gly Lys Val Ala Phe Asp Ile Trp 
        115                 120                 125             


Gly Gln Gly Thr Met Val Thr Val Ser Ser 
    130                 135             


<210> 4
<211> 133
<212> PRT
<213> Homo sapiens

<400> 4
Met Gly Thr Pro Ala Gln Leu Leu Phe Leu Leu Leu Leu Trp Leu Pro 
1               5                   10                  15      


Asp Thr Thr Gly Asp Ile Val Met Thr Gln Ser Pro Asp Ser Leu Ala 
            20                  25                  30          


Val Ser Leu Gly Glu Arg Ala Thr Ile Asn Cys Lys Ser Ser Gln Ser 
        35                  40                  45              


Val Leu Tyr Ser Pro Asn Asn Lys Asn Tyr Leu Ala Trp Tyr Gln Gln 
    50                  55                  60                  


Lys Pro Gly Gln Pro Pro Lys Leu Leu Ile Tyr Trp Ala Ser Thr Arg 
65                  70                  75                  80  


Glu Ser Gly Val Pro Asp Arg Phe Ser Gly Ser Gly Ser Gly Thr Asp 
                85                  90                  95      


Phe Thr Leu Thr Ile Ser Ser Leu Gln Ala Glu Asp Val Ala Val Tyr 
            100                 105                 110         


Tyr Cys Gln Gln Tyr Tyr Gly Ser Pro Ile Thr Phe Gly Gly Gly Thr 
        115                 120                 125             


Lys Val Glu Ile Lys 
    130             


<210> 5
<211> 142
<212> PRT
<213> Homo sapiens

<400> 5
Met Gly Phe Gly Leu Ser Trp Leu Phe Leu Val Ala Ile Leu Lys Gly 
1               5                   10                  15      


Val Gln Cys Gln Val Gln Leu Val Gln Ser Gly Ala Glu Val Lys Lys 
            20                  25                  30          


Pro Gly Ala Ser Val Lys Val Ser Cys Lys Ala Ser Gly Tyr Ala Phe 
        35                  40                  45              


Thr Ser Tyr Gly Ile Asn Trp Val Arg Gln Ala Pro Gly Gln Gly Leu 
    50                  55                  60                  


Glu Trp Met Gly Trp Ile Ser Ala Tyr Asn Gly Asn Thr Tyr Tyr Ala 
65                  70                  75                  80  


Gln Lys Leu Arg Gly Arg Val Thr Met Thr Thr Asp Thr Ser Thr Ser 
                85                  90                  95      


Thr Ala Tyr Met Glu Leu Arg Ser Leu Arg Ser Asp Asp Thr Ala Val 
            100                 105                 110         


Tyr Tyr Cys Ala Arg Asp Leu Gly Gly Tyr Gly Ser Gly Ser Val Pro 
        115                 120                 125             


Phe Asp Pro Trp Gly Gln Gly Thr Leu Val Thr Val Ser Ser 
    130                 135                 140         


<210> 6
<211> 128
<212> PRT
<213> Homo sapiens

<400> 6
Met Gly Thr Pro Ala Gln Leu Leu Phe Leu Leu Leu Leu Trp Leu Pro 
1               5                   10                  15      


Asp Thr Thr Gly Glu Ile Val Met Thr Gln Ser Pro Ala Thr Leu Ser 
            20                  25                  30          


Val Ser Pro Gly Glu Arg Ala Thr Leu Ser Cys Arg Ala Ser Gln Ser 
        35                  40                  45              


Val Ser Ser Asn Leu Ala Trp Tyr Gln Gln Lys Pro Gly Gln Ala Pro 
    50                  55                  60                  


Arg Leu Leu Ile Tyr Gly Ala Ser Thr Arg Ala Thr Gly Ile Pro Ala 
65                  70                  75                  80  


Arg Phe Ser Gly Ser Gly Ser Gly Thr Glu Phe Thr Leu Thr Ile Ser 
                85                  90                  95      


Ser Leu Gln Ser Glu Asp Phe Ala Val Tyr Tyr Cys Gln Asp Tyr Arg 
            100                 105                 110         


Thr Trp Pro Arg Arg Val Phe Gly Gly Gly Thr Lys Val Glu Ile Lys 
        115                 120                 125             


<210> 7
<211> 5
<212> PRT
<213> Homo sapiens

<400> 7
Ser Tyr Ala Ile Ser 
1               5   


<210> 8
<211> 10
<212> PRT
<213> Homo sapiens

<400> 8
Ile Ile Pro Ile Phe Gly Thr Val Asn Tyr 
1               5                   10  


<210> 9
<211> 6
<212> PRT
<213> Homo sapiens

<400> 9
Asp Pro Ser Val Asn Leu 
1               5       


<210> 10
<211> 8
<212> PRT
<213> Homo sapiens

<400> 10
Gln Ser Ile Ser Ser Trp Trp Ala 
1               5               


<210> 11
<211> 5
<212> PRT
<213> Homo sapiens

<400> 11
Asp Ala Ser Ser Leu 
1               5   


<210> 12
<211> 7
<212> PRT
<213> Homo sapiens

<400> 12
Gln Gln Tyr His Ala His Pro 
1               5           


<210> 13
<211> 5
<212> PRT
<213> Homo sapiens

<400> 13
Ser Tyr Ala Ile Ser 
1               5   


<210> 14
<211> 10
<212> PRT
<213> Homo sapiens

<400> 14
Ile Ile Pro Ile Phe Gly Ala Ala Asn Pro 
1               5                   10  


<210> 15
<211> 6
<212> PRT
<213> Homo sapiens

<400> 15
Met Gly Arg Gly Lys Val 
1               5       


<210> 16
<211> 14
<212> PRT
<213> Homo sapiens

<400> 16
Gln Ser Val Leu Tyr Ser Pro Asn Asn Lys Asn Tyr Leu Ala 
1               5                   10                  


<210> 17
<211> 5
<212> PRT
<213> Homo sapiens

<400> 17
Trp Ala Ser Thr Arg 
1               5   


<210> 18
<211> 7
<212> PRT
<213> Homo sapiens

<400> 18
Gln Gln Tyr Tyr Gly Ser Pro 
1               5           


<210> 19
<211> 5
<212> PRT
<213> Homo sapiens

<400> 19
Ser Tyr Gly Ile Asn 
1               5   


<210> 20
<211> 10
<212> PRT
<213> Homo sapiens

<400> 20
Ile Ser Ala Tyr Asn Gly Asn Thr Tyr Tyr 
1               5                   10  


<210> 21
<211> 9
<212> PRT
<213> Homo sapiens

<400> 21
Asp Leu Gly Gly Tyr Gly Ser Gly Ser 
1               5                   


<210> 22
<211> 8
<212> PRT
<213> Homo sapiens

<400> 22
Gln Ser Val Ser Ser Asn Leu Ala 
1               5               


<210> 23
<211> 5
<212> PRT
<213> Homo sapiens

<400> 23
Gly Ala Ser Thr Arg 
1               5   


<210> 24
<211> 8
<212> PRT
<213> Homo sapiens

<400> 24
Gln Asp Tyr Arg Thr Trp Pro Arg 
1               5               


