                         SEQUENCE LISTING

<110>  New York University
 
<120>  OSTEOPONTIN ISOFORM A INHIBITORS AND METHODS OF USE

<130>  29527.1241

<150>  61/598,115
<151>  2012-02-13

<160>  23    

<170>  PatentIn version 3.5

<210>  1
<211>  1641
<212>  DNA
<213>  Homo sapiens

<400>  1
ctccctgtgt tggtggagga tgtctgcagc agcatttaaa ttctgggagg gcttggttgt       60

cagcagcagc aggaggaggc agagcacagc atcgtcggga ccagactcgt ctcaggccag      120

ttgcagcctt ctcagccaaa cgccgaccaa ggaaaactca ctaccatgag aattgcagtg      180

atttgctttt gcctcctagg catcacctgt gccataccag ttaaacaggc tgattctgga      240

agttctgagg aaaagcagct ttacaacaaa tacccagatg ctgtggccac atggctaaac      300

cctgacccat ctcagaagca gaatctccta gccccacaga atgctgtgtc ctctgaagaa      360

accaatgact ttaaacaaga gacccttcca agtaagtcca acgaaagcca tgaccacatg      420

gatgatatgg atgatgaaga tgatgatgac catgtggaca gccaggactc cattgactcg      480

aacgactctg atgatgtaga tgacactgat gattctcacc agtctgatga gtctcaccat      540

tctgatgaat ctgatgaact ggtcactgat tttcccacgg acctgccagc aaccgaagtt      600

ttcactccag ttgtccccac agtagacaca tatgatggcc gaggtgatag tgtggtttat      660

ggactgaggt caaaatctaa gaagtttcgc agacctgaca tccagtaccc tgatgctaca      720

gacgaggaca tcacctcaca catggaaagc gaggagttga atggtgcata caaggccatc      780

cccgttgccc aggacctgaa cgcgccttct gattgggaca gccgtgggaa ggacagttat      840

gaaacgagtc agctggatga ccagagtgct gaaacccaca gccacaagca gtccagatta      900

tataagcgga aagccaatga tgagagcaat gagcattccg atgtgattga tagtcaggaa      960

ctttccaaag tcagccgtga attccacagc catgaatttc acagccatga agatatgctg     1020

gttgtagacc ccaaaagtaa ggaagaagat aaacacctga aatttcgtat ttctcatgaa     1080

ttagatagtg catcttctga ggtcaattaa aaggagaaaa aatacaattt ctcactttgc     1140

atttagtcaa aagaaaaaat gctttatagc aaaatgaaag agaacatgaa atgcttcttt     1200

ctcagtttat tggttgaatg tgtatctatt tgagtctgga aataactaat gtgtttgata     1260

attagtttag tttgtggctt catggaaact ccctgtaaac taaaagcttc agggttatgt     1320

ctatgttcat tctatagaag aaatgcaaac tatcactgta ttttaatatt tgttattctc     1380

tcatgaatag aaatttatgt agaagcaaac aaaatacttt tacccactta aaaagagaat     1440

ataacatttt atgtcactat aatcttttgt tttttaagtt agtgtatatt ttgttgtgat     1500

tatctttttg tggtgtgaat aaatctttta tcttgaatgt aataagaatt tggtggtgtc     1560

aattgcttat ttgttttccc acggttgtcc agcaattaat aaaacataac cttttttact     1620

gcctaaaaaa aaaaaaaaaa a                                               1641


<210>  2
<211>  314
<212>  PRT
<213>  Homo sapiens

<400>  2

Met Arg Ile Ala Val Ile Cys Phe Cys Leu Leu Gly Ile Thr Cys Ala 
1               5                   10                  15      


Ile Pro Val Lys Gln Ala Asp Ser Gly Ser Ser Glu Glu Lys Gln Leu 
            20                  25                  30          


Tyr Asn Lys Tyr Pro Asp Ala Val Ala Thr Trp Leu Asn Pro Asp Pro 
        35                  40                  45              


Ser Gln Lys Gln Asn Leu Leu Ala Pro Gln Asn Ala Val Ser Ser Glu 
    50                  55                  60                  


Glu Thr Asn Asp Phe Lys Gln Glu Thr Leu Pro Ser Lys Ser Asn Glu 
65                  70                  75                  80  


Ser His Asp His Met Asp Asp Met Asp Asp Glu Asp Asp Asp Asp His 
                85                  90                  95      


Val Asp Ser Gln Asp Ser Ile Asp Ser Asn Asp Ser Asp Asp Val Asp 
            100                 105                 110         


Asp Thr Asp Asp Ser His Gln Ser Asp Glu Ser His His Ser Asp Glu 
        115                 120                 125             


Ser Asp Glu Leu Val Thr Asp Phe Pro Thr Asp Leu Pro Ala Thr Glu 
    130                 135                 140                 


Val Phe Thr Pro Val Val Pro Thr Val Asp Thr Tyr Asp Gly Arg Gly 
145                 150                 155                 160 


Asp Ser Val Val Tyr Gly Leu Arg Ser Lys Ser Lys Lys Phe Arg Arg 
                165                 170                 175     


Pro Asp Ile Gln Tyr Pro Asp Ala Thr Asp Glu Asp Ile Thr Ser His 
            180                 185                 190         


Met Glu Ser Glu Glu Leu Asn Gly Ala Tyr Lys Ala Ile Pro Val Ala 
        195                 200                 205             


Gln Asp Leu Asn Ala Pro Ser Asp Trp Asp Ser Arg Gly Lys Asp Ser 
    210                 215                 220                 


Tyr Glu Thr Ser Gln Leu Asp Asp Gln Ser Ala Glu Thr His Ser His 
225                 230                 235                 240 


Lys Gln Ser Arg Leu Tyr Lys Arg Lys Ala Asn Asp Glu Ser Asn Glu 
                245                 250                 255     


His Ser Asp Val Ile Asp Ser Gln Glu Leu Ser Lys Val Ser Arg Glu 
            260                 265                 270         


Phe His Ser His Glu Phe His Ser His Glu Asp Met Leu Val Val Asp 
        275                 280                 285             


Pro Lys Ser Lys Glu Glu Asp Lys His Leu Lys Phe Arg Ile Ser His 
    290                 295                 300                 


Glu Leu Asp Ser Ala Ser Ser Glu Val Asn 
305                 310                 


<210>  3
<211>  27
<212>  PRT
<213>  Artificial

<220>
<223>  Peptide mimic of OPNa exon 4

<400>  3

Leu Tyr Asn Lys Tyr Pro Asp Ala Val Ala Thr Trp Leu Asn Pro Asp 
1               5                   10                  15      


Pro Ser Gln Lys Gln Asn Leu Leu Ala Pro Gln 
            20                  25          


<210>  4
<211>  17
<212>  PRT
<213>  Artificial

<220>
<223>  Peptide mimic of OPNa exon 4

<400>  4

Lys Tyr Pro Asp Ala Val Ala Thr Trp Leu Asn Pro Asp Pro Ser Gln 
1               5                   10                  15      


Lys 
    


<210>  5
<211>  4
<212>  PRT
<213>  Artificial

<220>
<223>  R2 of peptide mimic of OPNa exon 4

<400>  5

Pro Asp Ala Val 
1               


<210>  6
<211>  4
<212>  PRT
<213>  Artificial

<220>
<223>  R1 of peptide mimic of OPNa exon 4

<400>  6

Tyr Asn Lys Tyr 
1               


<210>  7
<211>  5
<212>  PRT
<213>  Artificial

<220>
<223>  R1 of peptide mimic of OPNa exon 4

<400>  7

Leu Tyr Asn Lys Tyr 
1               5   


<210>  8
<211>  4
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  8

Ala Thr Trp Leu 
1               


<210>  9
<211>  5
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  9

Ala Thr Trp Leu Asn 
1               5   


<210>  10
<211>  6
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  10

Ala Thr Trp Leu Asn Pro 
1               5       


<210>  11
<211>  7
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  11

Ala Thr Trp Leu Asn Pro Asp 
1               5           


<210>  12
<211>  8
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  12

Ala Thr Trp Leu Asn Pro Asp Pro 
1               5               


<210>  13
<211>  9
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  13

Ala Thr Trp Leu Asn Pro Asp Pro Ser 
1               5                   


<210>  14
<211>  10
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  14

Ala Thr Trp Leu Asn Pro Asp Pro Ser Gln 
1               5                   10  


<210>  15
<211>  11
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  15

Ala Thr Trp Leu Asn Pro Asp Pro Ser Gln Lys 
1               5                   10      


<210>  16
<211>  12
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  16

Ala Thr Trp Leu Asn Pro Asp Pro Ser Gln Lys Gln 
1               5                   10          


<210>  17
<211>  13
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  17

Ala Thr Trp Leu Asn Pro Asp Pro Ser Gln Lys Gln Asn 
1               5                   10              


<210>  18
<211>  14
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  18

Ala Thr Trp Leu Asn Pro Asp Pro Ser Gln Lys Gln Asn Leu 
1               5                   10                  


<210>  19
<211>  15
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  19

Ala Thr Trp Leu Asn Pro Asp Pro Ser Gln Lys Gln Asn Leu Leu 
1               5                   10                  15  


<210>  20
<211>  16
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  20

Ala Thr Trp Leu Asn Pro Asp Pro Ser Gln Lys Gln Asn Leu Leu Ala 
1               5                   10                  15      


<210>  21
<211>  17
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  21

Ala Thr Trp Leu Asn Pro Asp Pro Ser Gln Lys Gln Asn Leu Leu Ala 
1               5                   10                  15      


Pro 
    


<210>  22
<211>  18
<212>  PRT
<213>  Artificial

<220>
<223>  R3 of peptide mimic of OPNa exon 4

<400>  22

Ala Thr Trp Leu Asn Pro Asp Pro Ser Gln Lys Gln Asn Leu Leu Ala 
1               5                   10                  15      


Pro Gln 
        


<210>  23
<211>  17
<212>  PRT
<213>  Artificial

<220>
<223>  Scrambled Sham Peptide

<400>  23

Trp Gln Lys Pro Ala Pro Leu Asp Thr Asp Pro Lys Val Tyr Ala Asn 
1               5                   10                  15      


Ser 
    


