                         SEQUENCE LISTING

<110>  Bayer Schering Pharma AG
 
<120>  Modulators of SLC22A7

<130>  BHC 10 1 048

<160>  13    

<170>  PatentIn version 3.5

<210>  1
<211>  2136
<212>  DNA
<213>  Homo sapiens

<400>  1
ccacctccag agtccaaggg tctatgtggt gggcagtttg agctggctgg atactagagg       60

gaggctgcac ctgaagcatt tggtgggtga gcagcatggg ctttgaggag ctgctggagc      120

aggtgggcgg ctttgggccc ttccaactgc ggaatgtggc actgctggcc ctgccccgag      180

tgctgctacc actgcacttc ctcctgccca tcttcctggc tgccgtgcct gcccaccgat      240

gtgccctgcc gggtgcccct gccaacttca gccatcagga tgtgtggctg gaggcccatc      300

ttccccggga gcctgatggc acgctcagct cctgcctccg ctttgcctat ccccaggctc      360

tccccaacac cacgttgggg gaagaaaggc agagccgtgg ggagctggag gatgaacctg      420

ccacagtgcc ctgctctcag ggctgggagt acgaccactc agaattctcc tctaccattg      480

caactgagtc ccagtgggat ctggtgtgtg agcagaaagg tctgaacaga gctgcgtcca      540

ctttcttctt cgccggtgtg ctggtggggg ctgtggcctt tggatatctg tccgacaggt      600

ttgggcggcg gcgtctgctg ctggtagcct acgtgagtac cctggtgctg ggcctggcat      660

ctgcagcctc cgtcagctat gtaatgtttg ccatcacccg cacccttact ggctcagccc      720

tggctggttt taccatcatc gtgatgccac tggagctgga gtggctggat gtggagcacc      780

gcaccgtggc tggagtcctg agcagcacct tctggacagg gggcgtgatg ctgctggcac      840

tggttgggta cctgatacgg gactggcgat ggcttctgct agctgtcacc ctgccttgtg      900

ccccaggcat cctcagcctc tggtgggtgc ctgagtctgc acgctggctt ctgacccaag      960

gccatgtgaa agaggcccac aggtacttgc tccactgtgc caggctcaat gggcggccag     1020

tgtgtgagga cagcttcagc caggaggctg tgagcaaagt ggccgccggg gaacgggtgg     1080

tccgaagacc ttcataccta gacctgttcc gcacaccacg gctccgacac atctcactgt     1140

gctgcgtggt ggtgtggttc ggagtgaact tctcctatta cggcctgagt ctggatgtgt     1200

cggggctggg gctgaacgtg taccagacac agctgttgtt cggggctgtg gaactgccct     1260

ccaagctgct ggtctacttg tcggtgcgct acgcaggacg ccgcctcacg caagccggga     1320

cactgctggg cacggccctg gcgttcggca ctagactgct agtgtcctcc gatatgaagt     1380

cctggagcac tgtcctggca gtgatgggga aagctttttc tgaagctgcc ttcaccactg     1440

cttacctgtt cacttcagag ttgtacccta cggtgctcag acagacaggg atggggctga     1500

ctgcactggt gggccggctg gggggctctt tggccccact ggcggccttg ctagatggag     1560

tgtggctgtc actgcccaag cttacttatg gggggatcgc cctgctggct gccggcaccg     1620

ccctcctgct gccagagacg aggcaggcac agctgccaga gaccatccag gacgtggaga     1680

gaaagagtgc cccaaccagt cttcaggagg aagagatgcc catgaagcag gtccagaact     1740

aagtgggagt ggaggcaggc cctccacaga agctctgcag caggggctgg gagagcagaa     1800

gggcaggccc ttcaactcag gctgggagag cagaagggca ggccctgcaa ctcaggctgg     1860

gagtatcgaa ccctctgcct agggccggag ttgctgccag tacccgctcc ctctgctcat     1920

ccatccttga ttatttggct tctaggaaca gttgacttcc cagaatgcag tgggctgctg     1980

ggcacccctc tcacggttgg ggaggattct gtaaataaag gtgccccttg ggttggggca     2040

gtggtgacga gctgtgggaa gagccctgga taggaagcca ctgagtctgc cctgggctct     2100

gataaaactt caccattaaa aaaaaaaaaa aaaaaa                               2136


<210>  2
<211>  548
<212>  PRT
<213>  Homo sapiens

<400>  2

Met Gly Phe Glu Glu Leu Leu Glu Gln Val Gly Gly Phe Gly Pro Phe 
1               5                   10                  15      


Gln Leu Arg Asn Val Ala Leu Leu Ala Leu Pro Arg Val Leu Leu Pro 
            20                  25                  30          


Leu His Phe Leu Leu Pro Ile Phe Leu Ala Ala Val Pro Ala His Arg 
        35                  40                  45              


Cys Ala Leu Pro Gly Ala Pro Ala Asn Phe Ser His Gln Asp Val Trp 
    50                  55                  60                  


Leu Glu Ala His Leu Pro Arg Glu Pro Asp Gly Thr Leu Ser Ser Cys 
65                  70                  75                  80  


Leu Arg Phe Ala Tyr Pro Gln Ala Leu Pro Asn Thr Thr Leu Gly Glu 
                85                  90                  95      


Glu Arg Gln Ser Arg Gly Glu Leu Glu Asp Glu Pro Ala Thr Val Pro 
            100                 105                 110         


Cys Ser Gln Gly Trp Glu Tyr Asp His Ser Glu Phe Ser Ser Thr Ile 
        115                 120                 125             


Ala Thr Glu Ser Gln Trp Asp Leu Val Cys Glu Gln Lys Gly Leu Asn 
    130                 135                 140                 


Arg Ala Ala Ser Thr Phe Phe Phe Ala Gly Val Leu Val Gly Ala Val 
145                 150                 155                 160 


Ala Phe Gly Tyr Leu Ser Asp Arg Phe Gly Arg Arg Arg Leu Leu Leu 
                165                 170                 175     


Val Ala Tyr Val Ser Thr Leu Val Leu Gly Leu Ala Ser Ala Ala Ser 
            180                 185                 190         


Val Ser Tyr Val Met Phe Ala Ile Thr Arg Thr Leu Thr Gly Ser Ala 
        195                 200                 205             


Leu Ala Gly Phe Thr Ile Ile Val Met Pro Leu Glu Leu Glu Trp Leu 
    210                 215                 220                 


Asp Val Glu His Arg Thr Val Ala Gly Val Leu Ser Ser Thr Phe Trp 
225                 230                 235                 240 


Thr Gly Gly Val Met Leu Leu Ala Leu Val Gly Tyr Leu Ile Arg Asp 
                245                 250                 255     


Trp Arg Trp Leu Leu Leu Ala Val Thr Leu Pro Cys Ala Pro Gly Ile 
            260                 265                 270         


Leu Ser Leu Trp Trp Val Pro Glu Ser Ala Arg Trp Leu Leu Thr Gln 
        275                 280                 285             


Gly His Val Lys Glu Ala His Arg Tyr Leu Leu His Cys Ala Arg Leu 
    290                 295                 300                 


Asn Gly Arg Pro Val Cys Glu Asp Ser Phe Ser Gln Glu Ala Val Ser 
305                 310                 315                 320 


Lys Val Ala Ala Gly Glu Arg Val Val Arg Arg Pro Ser Tyr Leu Asp 
                325                 330                 335     


Leu Phe Arg Thr Pro Arg Leu Arg His Ile Ser Leu Cys Cys Val Val 
            340                 345                 350         


Val Trp Phe Gly Val Asn Phe Ser Tyr Tyr Gly Leu Ser Leu Asp Val 
        355                 360                 365             


Ser Gly Leu Gly Leu Asn Val Tyr Gln Thr Gln Leu Leu Phe Gly Ala 
    370                 375                 380                 


Val Glu Leu Pro Ser Lys Leu Leu Val Tyr Leu Ser Val Arg Tyr Ala 
385                 390                 395                 400 


Gly Arg Arg Leu Thr Gln Ala Gly Thr Leu Leu Gly Thr Ala Leu Ala 
                405                 410                 415     


Phe Gly Thr Arg Leu Leu Val Ser Ser Asp Met Lys Ser Trp Ser Thr 
            420                 425                 430         


Val Leu Ala Val Met Gly Lys Ala Phe Ser Glu Ala Ala Phe Thr Thr 
        435                 440                 445             


Ala Tyr Leu Phe Thr Ser Glu Leu Tyr Pro Thr Val Leu Arg Gln Thr 
    450                 455                 460                 


Gly Met Gly Leu Thr Ala Leu Val Gly Arg Leu Gly Gly Ser Leu Ala 
465                 470                 475                 480 


Pro Leu Ala Ala Leu Leu Asp Gly Val Trp Leu Ser Leu Pro Lys Leu 
                485                 490                 495     


Thr Tyr Gly Gly Ile Ala Leu Leu Ala Ala Gly Thr Ala Leu Leu Leu 
            500                 505                 510         


Pro Glu Thr Arg Gln Ala Gln Leu Pro Glu Thr Ile Gln Asp Val Glu 
        515                 520                 525             


Arg Lys Ser Ala Pro Thr Ser Leu Gln Glu Glu Glu Met Pro Met Lys 
    530                 535                 540                 


Gln Val Gln Asn 
545             


<210>  3
<211>  37
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  primer

<400>  3

Gly Thr Thr Thr Ala Ala Ala Cys Thr Thr Ala Ala Gly Cys Thr Thr 
1               5                   10                  15      


Gly Cys Cys Ala Cys Cys Ala Thr Gly Gly Gly Cys Thr Thr Thr Gly 
            20                  25                  30          


Ala Gly Gly Ala Gly 
        35          


<210>  4
<211>  25
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  primer

<400>  4
gtccagaact aactcgagcg atcgc                                             25


<210>  5
<211>  37
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  primer

<400>  5
gtttaaactt aagcttgcca ccatgggctt cgaagac                                37


<210>  6
<211>  25
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  primer

<400>  6
cttcccgcag cactcgagcg atcgc                                             25


<210>  7
<211>  37
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  primer

<400>  7
gtttaaactt aagcttgcca ccatggcctt taatgac                                37


<210>  8
<211>  25
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  primer

<400>  8
aatggactct gactcgagcg atcgc                                             25


<210>  9
<211>  37
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  primer

<400>  9
gtttaaactt aagcttgcca ccatggctca gtttgtc                                37


<210>  10
<211>  25
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  primer

<400>  10
aagagctgga ccctcgagcg atcgc                                             25


<210>  11
<211>  21
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  primer

<400>  11
ctgtggcctt tggatatctg t                                                 21


<210>  12
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  primer

<400>  12
acgtaggcta ccagcagcag                                                   20


<210>  13
<211>  18
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  primer

<400>  13
cgacaggttt gggcggcg                                                     18


