                         SEQUENCE LISTING

<110>  RXi Pharmaceuticals Corporation
       BULOCK, Karen
       KHVOROVA, Anastasia
       LAPIERRE, Jennifer
 
<120>  FORMULATIONS AND METHODS FOR TARGETED DELIVERY TO PHAGOCTYE CELLS

<130>  R0659.70017WO00

<150>  US 61/310,611
<151>  2010-03-04

<160>  19    

<170>  PatentIn version 3.5

<210>  1
<211>  80
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic Polypeptide

<400>  1

Lys Lys Lys Lys His His His Lys His His His Lys His His His Lys 
1               5                   10                  15      


His His His Lys His Lys His His His Lys His His His Lys His His 
            20                  25                  30          


His Lys His His His Lys His Lys His His His Lys His His His Lys 
        35                  40                  45              


His His His Lys His His His Lys His Lys His His His Lys His His 
    50                  55                  60                  


His Lys His His His Lys His His His Lys His His His His His Asn 
65                  70                  75                  80  


<210>  2
<211>  28
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic Polypeptide

<400>  2

Lys Glu Thr Trp Trp Glu Thr Trp Trp Thr Glu Trp Ser Gln Pro Gly 
1               5                   10                  15      


Arg Lys Lys Arg Arg Gln Arg Arg Arg Pro Pro Gln 
            20                  25              


<210>  3
<211>  36
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic Polypeptide

<400>  3

Lys Gly Ser Lys Lys Ala Val Thr Lys Ala Gln Lys Lys Asp Gly Lys 
1               5                   10                  15      


Lys Arg Lys Arg Ser Arg Lys Glu Ser Tyr Ser Val Tyr Val Tyr Lys 
            20                  25                  30          


Val Leu Lys Gln 
        35      


<210>  4
<211>  13
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  DY547 attached

<220>
<221>  misc_feature
<222>  (1)..(2)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (4)..(4)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (10)..(12)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (13)..(13)
<223>  cholesterol attached

<400>  4
cuguggaagu cua                                                          13


<210>  5
<211>  19
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  5'-Phosphate

<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  2'-Fluoro

<220>
<221>  misc_feature
<222>  (5)..(9)
<223>  2'-Fluoro

<220>
<221>  misc_feature
<222>  (11)..(11)
<223>  2'-Fluoro

<220>
<221>  misc_feature
<222>  (11)..(19)
<223>  phosphorothioate linkage

<220>
<221>  misc_feature
<222>  (14)..(17)
<223>  2'-Fluoro

<400>  5
uagacuucca cagucucaa                                                    19


<210>  6
<211>  13
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  DY547 attached

<220>
<221>  misc_feature
<222>  (1)..(2)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (4)..(4)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (10)..(12)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (13)..(13)
<223>  cholesterol attached

<400>  6
cuguggaagu cua                                                          13


<210>  7
<211>  19
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  5'-Phosphate

<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  2'-Fluoro

<220>
<221>  misc_feature
<222>  (5)..(9)
<223>  2'-Fluoro

<220>
<221>  misc_feature
<222>  (11)..(11)
<223>  2'-Fluoro

<220>
<221>  misc_feature
<222>  (11)..(19)
<223>  phosphorothioate linkage

<220>
<221>  misc_feature
<222>  (16)..(18)
<223>  2'-Fluoro

<400>  7
uagacuucca cagaacucu                                                    19


<210>  8
<211>  13
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(2)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (4)..(4)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (10)..(12)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (13)..(13)
<223>  cholesterol attached

<400>  8
cuguggaagu cua                                                          13


<210>  9
<211>  19
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  5'-Phosphate

<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (5)..(9)
<223>  2'-Fluoro

<220>
<221>  misc_feature
<222>  (11)..(11)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (13)..(19)
<223>  phosphorothioate linkage

<220>
<221>  misc_feature
<222>  (16)..(18)
<223>  2'-O-methyl

<400>  9
uagacuucca cagaacucu                                                    19


<210>  10
<211>  13
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  DY547 attached

<220>
<221>  misc_feature
<222>  (1)..(2)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (4)..(4)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (10)..(12)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (13)..(13)
<223>  cholesterol attached

<400>  10
cuguggaagu cua                                                          13


<210>  11
<211>  19
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  5'-Phosphate

<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (5)..(9)
<223>  2'-Fluoro

<220>
<221>  misc_feature
<222>  (11)..(11)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (13)..(19)
<223>  phosphorothioate linkage

<220>
<221>  misc_feature
<222>  (16)..(18)
<223>  2'-O-methyl

<400>  11
uagacuucca cagaacucu                                                    19


<210>  12
<211>  13
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  DY547 attached

<220>
<221>  misc_feature
<222>  (2)..(2)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (6)..(6)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (8)..(8)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (11)..(13)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (13)..(13)
<223>  cholesterol attached

<400>  12
acaaauacga uuu                                                          13


<210>  13
<211>  19
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  5'-Phosphate

<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (4)..(5)
<223>  2'-Fluoro

<220>
<221>  misc_feature
<222>  (7)..(7)
<223>  2'-Fluoro

<220>
<221>  misc_feature
<222>  (9)..(10)
<223>  2'-Fluoro

<220>
<221>  misc_feature
<222>  (11)..(11)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (13)..(14)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (13)..(19)
<223>  phosphorothioate linkage

<220>
<221>  misc_feature
<222>  (17)..(18)
<223>  2'-O-methyl

<400>  13
aaaucguauu ugucaauca                                                    19


<210>  14
<211>  25
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(1)
<223>  Cy3 attached

<220>
<221>  misc_feature
<222>  (1)..(12)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (16)..(25)
<223>  2'-O-methyl

<400>  14
cucuucggaa agacuguucc aaaaa                                             25


<210>  15
<211>  25
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide

<400>  15
uuuuuggaac agucuuuccg aagag                                             25


<210>  16
<211>  25
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(12)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (16)..(25)
<223>  2'-O-methyl

<400>  16
gaggguuaac ggugugucac cauga                                             25


<210>  17
<211>  25
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide

<400>  17
ucauggugac acaccguuaa cccuc                                             25


<210>  18
<211>  25
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide


<220>
<221>  misc_feature
<222>  (1)..(12)
<223>  2'-O-methyl

<220>
<221>  misc_feature
<222>  (16)..(25)
<223>  2'-O-methyl

<400>  18
cucuucggaa agacuguucc aaaaa                                             25


<210>  19
<211>  25
<212>  RNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Oligonucleotide

<400>  19
uuuuuggaac agucuuuccg aagag                                             25


