(WO/2006/091974) TADALAFIL HAVING A LARGE PARTICLE SIZE AND A PROCESS FOR PREPARATION THEREOF
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| Latest bibliographic data on file with the International Bureau
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| Pub. No.: | WO/2006/091974 | International Application No.: | PCT/US2006/007076 | |||
| Publication Date: | 31.08.2006 | International Filing Date: | 27.02.2006 |
| IPC: | C07D 471/14 (2006.01), A61K 31/4985 (2006.01) | |||||||||||||||||||||||||||||||||||
| Applicants: | TEVA PHARMACEUTICAL INDUSTRIES LTD. [IL/IL]; 5 BASEL STREET, P.O. Box 3190, 49131 Petah Tiqva (IL) (AE, AG, AL, AM, AT, AU, AZ, BA, BE, BF, BG, BJ, BR, BW, BY, BZ, CA, CF, CG, CH, CI, CM, CN, CO, CR, CU, CY, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, FR, GA, GB, GD, GE, GH, GM, GN, GQ, GR, GW, HR, HU, ID, IE, IL, IN, IS, IT, JP, KE, KG, KM, KN, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, LY, MA, MC, MD, MG, MK, ML, MN, MR, MW, MX, MZ, NA, NE, NG, NI, NL, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SI, SK, SL, SM, SN, SY, SZ, TD, TG, TJ, TM, TN, TR, TT, TZ, UA, UG, UZ, VC, VN, YU, ZA, ZM, ZW only). TEVA PHARMACEUTICALS USA INC. [US/US]; 1090 HORSHAM ROAD, P.O. Box 1090, North Wales, PA 19454 (US) (BB only). ORNAN, Inbal [IL/IL]; (IL) (US Only). AMIR, Ehud [IL/IL]; (IL) (US Only). SAMBURSKI, Guy [IL/IL]; (IL) (US Only). OVADYA, Yhoshoa [IL/IL]; (IL) (US Only). | |||||||||||||||||||||||||||||||||||
| Inventors: | ORNAN, Inbal; (IL). AMIR, Ehud; (IL). SAMBURSKI, Guy; (IL). OVADYA, Yhoshoa; (IL). | |||||||||||||||||||||||||||||||||||
| Agent: | BRAINARD, Charles, R. et al.; KENYON & KENYON LLP, One Broadway, New York, NY 10004-1050 (US) . | |||||||||||||||||||||||||||||||||||
| Priority Data: |
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| Title: | TADALAFIL HAVING A LARGE PARTICLE SIZE AND A PROCESS FOR PREPARATION THEREOF | |||||||||||||||||||||||||||||||||||
| Abstract: | The present invention provides particulate tadalafil having a particle size of about 200 to about 600 microns and a process for controlling the particle size of tadalafil. | |||||||||||||||||||||||||||||||||||
| Designated States: |
AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW. African Regional Intellectual Property Org. (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW) Eurasian Patent Organization (EAPO) (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM) European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR) African Intellectual Property Organization (OAPI) (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG). |
| Publication Language: | English (EN) |
| Filing Language: | English (EN) |


