(WO/2006/091974) TADALAFIL HAVING A LARGE PARTICLE SIZE AND A PROCESS FOR PREPARATION THEREOF

(WO/2006/091974) TADALAFIL HAVING A LARGE PARTICLE SIZE AND A PROCESS FOR PREPARATION THEREOF

Latest bibliographic data on file with the International Bureau
Pub. No.:  WO/2006/091974   International Application No.:  PCT/US2006/007076
Publication Date:31.08.2006 International Filing Date:27.02.2006
IPC: C07D 471/14 (2006.01), A61K 31/4985 (2006.01)
Applicants:TEVA PHARMACEUTICAL INDUSTRIES LTD. [IL/IL]; 5 BASEL STREET, P.O. Box 3190, 49131 Petah Tiqva (IL) (AE, AG, AL, AM, AT, AU, AZ, BA, BE, BF, BG, BJ, BR, BW, BY, BZ, CA, CF, CG, CH, CI, CM, CN, CO, CR, CU, CY, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, FR, GA, GB, GD, GE, GH, GM, GN, GQ, GR, GW, HR, HU, ID, IE, IL, IN, IS, IT, JP, KE, KG, KM, KN, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, LY, MA, MC, MD, MG, MK, ML, MN, MR, MW, MX, MZ, NA, NE, NG, NI, NL, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SI, SK, SL, SM, SN, SY, SZ, TD, TG, TJ, TM, TN, TR, TT, TZ, UA, UG, UZ, VC, VN, YU, ZA, ZM, ZW only).
TEVA PHARMACEUTICALS USA INC. [US/US]; 1090 HORSHAM ROAD, P.O. Box 1090, North Wales, PA 19454 (US) (BB only).
ORNAN, Inbal [IL/IL]; (IL) (US Only).
AMIR, Ehud [IL/IL]; (IL) (US Only).
SAMBURSKI, Guy [IL/IL]; (IL) (US Only).
OVADYA, Yhoshoa [IL/IL]; (IL) (US Only).
Inventors:ORNAN, Inbal; (IL).
AMIR, Ehud; (IL).
SAMBURSKI, Guy; (IL).
OVADYA, Yhoshoa; (IL).
Agent:BRAINARD, Charles, R. et al.; KENYON & KENYON LLP, One Broadway, New York, NY 10004-1050 (US) .
Priority Data:
60/656,664 25.02.2005 US
60/677,514 03.05.2005 US
60/683,058 19.05.2005 US
60/733,012 02.11.2005 US
60/736,807 14.11.2005 US
60/737,080 15.11.2005 US
60/748,341 06.12.2005 US
Title: TADALAFIL HAVING A LARGE PARTICLE SIZE AND A PROCESS FOR PREPARATION THEREOF
Abstract: The present invention provides particulate tadalafil having a particle size of about 200 to about 600 microns and a process for controlling the particle size of tadalafil.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Org. (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (EAPO) (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (OAPI) (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language:English (EN)
Filing Language:English (EN)

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