(WO/2006/050458) TADALAFIL CRYSTAL FORMS AND PROCESSES FOR PREPARING THEM

(WO/2006/050458) TADALAFIL CRYSTAL FORMS AND PROCESSES FOR PREPARING THEM

Latest bibliographic data on file with the International Bureau
Pub. No.:  WO/2006/050458   International Application No.:  PCT/US2005/039828
Publication Date:11.05.2006 International Filing Date:02.11.2005
IPC: A61K 31/4985 (2006.01), A61P 15/10 (2006.01), C07D 471/14 (2006.01)
Applicants:TEVA PHARMACEUTICAL INDUSTRIES, LTD. [IL/IL]; 5 Basel Street, P.O. Box 3190, 49131 Petah Tiqva (IL) (AE, AG, AL, AM, AT, AU, AZ, BA, BE, BF, BG, BJ, BR, BW, BY, BZ, CA, CF, CG, CH, CI, CM, CN, CO, CR, CU, CY, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, FR, GA, GB, GD, GE, GH, GM, GN, GQ, GR, GW, HR, HU, ID, IE, IL, IN, IS, IT, JP, KE, KG, KM, KN, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, LY, MA, MC, MD, MG, MK, ML, MN, MR, MW, MX, MZ, NA, NE, NG, NI, NL, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SI, SK, SL, SM, SN, SY, SZ, TD, TG, TJ, TM, TN, TR, TT, TZ, UA, UG, UZ, VC, VN, YU, ZA, ZM, ZW only).
TEVA PHARMACEUTICALS USA, INC. [US/US]; 1090 Horsham Road, P.O Box 1090, North Wales, PA 19454 (US) (BB only).
WIZEL, Shlomit [IL/IL]; (IL) (US Only).
GIVANT, Ariel [IL/IL]; (IL) (US Only).
DILLER, Dov [IL/IL]; (IL) (US Only).
KROCHMAL, Barnaba [IL/IL]; (IL) (US Only).
Inventors:WIZEL, Shlomit; (IL).
GIVANT, Ariel; (IL).
DILLER, Dov; (IL).
KROCHMAL, Barnaba; (IL).
Agent:BRAINARD, CharleS, R. et al.; Kenyon & Kenyon, One Broadway, New York, NY 10004-1050 (US).
Priority Data:
60/624,412 02.11.2004 US
60/642,216 07.01.2005 US
Title: TADALAFIL CRYSTAL FORMS AND PROCESSES FOR PREPARING THEM
Abstract: The present invention provides tadalafil crystal forms II, III, IV, VI, VII, and VIII, and processes for preparing these forms. The present invention also provides processes for preparing tadalafil forms I and V.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Org. (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (EAPO) (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (OAPI) (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language:English (EN)
Filing Language:English (EN)

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