(WO/2002/018303) SYNTHESIS OF N,N-DIMETHYL-3-(4-METHYL) BENZOYL PROPIONAMIDE, A KEY INTERMEDIATE OF ZOLPIDEM

(WO/2002/018303) SYNTHESIS OF N,N-DIMETHYL-3-(4-METHYL) BENZOYL PROPIONAMIDE, A KEY INTERMEDIATE OF ZOLPIDEM

Latest bibliographic data on file with the International Bureau
Pub. No.:  WO/2002/018303   International Application No.:  PCT/IB2001/001558
Publication Date:07.03.2002 International Filing Date:28.08.2001
Chapter 2 Demand Filed: 21.03.2002
IPC: C07C 231/02 (2006.01), C07D 471/04 (2006.01), C07C 235/78 (2006.01)
Applicants:RANBAXY LABORATORIES LIMITED [IN/IN]; 19, Nehru Place, New Dehli 110 019, Maharashtra (IN) (All Except US).
KUMAR, Yatendra [IN/IN]; (IN) (US Only).
PRASAD, Mohan [IN/IN]; (IN) (US Only).
NATH, Asok [IN/IN]; (IN) (US Only).
Inventors:KUMAR, Yatendra; (IN).
PRASAD, Mohan; (IN).
NATH, Asok; (IN).
Common
Representative:
RANBAXY LABORATORIES LIMITED; DESHMUKH, Jayadeep, R., 600 College Road East, Suite 2100, Princeton, NJ 08540 (US).
Priority Data:
782/DEL/2000 29.08.2000 IN
Title: SYNTHESIS OF N,N-DIMETHYL-3-(4-METHYL) BENZOYL PROPIONAMIDE, A KEY INTERMEDIATE OF ZOLPIDEM
Abstract: The present invention relates to an improved and industrially advan-tageous process for the preparation of N, N-dimethyl-3-(4-methyl)benzoyl propionamide, which compound is a key intermediate for the synthesis of zolpidem hemitartrate, a non-benzodiazepine hypnotic agent.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NO, NZ, PH, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, TJ, TM, TR, TT, TZ, UA, UG, US, UZ, VN, YU, ZA, ZW.
African Regional Intellectual Property Org. (ARIPO) (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZW)
Eurasian Patent Organization (EAPO) (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE, TR)
African Intellectual Property Organization (OAPI) (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language:English (EN)
Filing Language:English (EN)

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