(WO/2009/006389) PYRIMIDINE DERIVATIVES USEFUL AS RAF KINASE INHIBITORS

(WO/2009/006389) PYRIMIDINE DERIVATIVES USEFUL AS RAF KINASE INHIBITORS

Latest bibliographic data on file with the International Bureau
Pub. No.:  WO/2009/006389   International Application No.:  PCT/US2008/068762
Publication Date:08.01.2009 International Filing Date:30.06.2008
IPC: C07D 401/12 (2006.01), A61K 31/506 (2006.01), A61P 29/00 (2006.01), A61P 35/00 (2006.01), C07D 401/14 (2006.01), C07D 403/12 (2006.01), C07D 413/14 (2006.01), C07D 417/12 (2006.01), C07D 417/14 (2006.01), C07D 471/04 (2006.01), C07D 473/00 (2006.01), C07D 487/04 (2006.01)
Applicants:SUNESIS PHARMACEUTICALS, INC. [US/US]; 395 Oyster Point Boulevard, Suite 400 South San Francisco, CA 94080 (US) (All Except US).
CHEN, Weirong [CN/US]; (US) (US Only).
COSSROW, Jennifer [US/US]; (US) (US Only).
FRANKLIN, Lioyd [US/US]; (US) (US Only).
GUAN, Bing [US/US]; (US) (US Only).
JONES, John, Howard [CA/US]; (US) (US Only).
KUMARAVEL, Gnanasambandam [US/US]; (US) (US Only).
LANE, Benjamin [US/US]; (US) (US Only).
LITTKE, Adam [CA/US]; (US) (US Only).
LUGOVSKOY, Alexey [RU/US]; (US) (US Only).
PENG, Hairuo [CN/US]; (US) (US Only).
POWELL, Noel [US/US]; (US) (US Only).
RAIMUNDO, Brian [US/US]; (US) (US Only).
TANAKA, Hiroko [JP/US]; (US) (US Only).
VESSELS, Jeffrey [US/US]; (US) (US Only).
WYNN, Thomas [US/US]; (US) (US Only).
XIN, Zhili [US/US]; (US) (US Only).
BIOGEN IDEC MA INC. [US/US]; 14 Cambridge Center Cambridge, MA 02142 (US) (All Except US).
Inventors:CHEN, Weirong; (US).
COSSROW, Jennifer; (US).
FRANKLIN, Lioyd; (US).
GUAN, Bing; (US).
JONES, John, Howard; (US).
KUMARAVEL, Gnanasambandam; (US).
LANE, Benjamin; (US).
LITTKE, Adam; (US).
LUGOVSKOY, Alexey; (US).
PENG, Hairuo; (US).
POWELL, Noel; (US).
RAIMUNDO, Brian; (US).
TANAKA, Hiroko; (US).
VESSELS, Jeffrey; (US).
WYNN, Thomas; (US).
XIN, Zhili; (US).
Agent:ROBIDOUX, Andrea, L.C.; Choate, Hall & Stewart LLP Two International Place Boston, MA 02110 (US).
Priority Data:
60/947,291 29.06.2007 US
Title: PYRIMIDINE DERIVATIVES USEFUL AS RAF KINASE INHIBITORS
Abstract: The present invention provides compounds useful as inhibitors of Raf protein kinase. The present invention also provides compositions thereof, and methods of treating Raf-mediated diseases.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Org. (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (EAPO) (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MT, NL, NO, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (OAPI) (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language:English (EN)
Filing Language:English (EN)

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