(WO/2008/124161) METHODS OF TREATING CANCER USING PYRIDOPYRIMIDINONE INHIBITORS OF PI3K ALPHA

(WO/2008/124161) METHODS OF TREATING CANCER USING PYRIDOPYRIMIDINONE INHIBITORS OF PI3K ALPHA

Latest bibliographic data on file with the International Bureau
Pub. No.:  WO/2008/124161   International Application No.:  PCT/US2008/004573
Publication Date:16.10.2008 International Filing Date:09.04.2008
IPC: A61K 31/517 (2006.01), A61K 31/282 (2006.01), A61K 31/337 (2006.01), A61K 31/4745 (2006.01), A61K 31/519 (2006.01), A61K 45/06 (2006.01), A61P 35/00 (2006.01)
Applicants:EXELIXIS, INC. [US/US]; 220 East Grand Avenue Post Office Box 511, South San Francisco, CA 94083 (US) (All Except US).
LAMB, Peter [US/US]; (US) (US Only).
MATTHEWS, David [GB/US]; (US) (US Only).
Inventors:LAMB, Peter; (US).
MATTHEWS, David; (US).
Agent:WADE, Janice V. et al.; EXELIXIS, Inc., 210 East Grand Avenue Post Office Box 511, South San Francisco, CA 94083-0511 (US).
Priority Data:
60/922,899 10.04.2007 US
Title: METHODS OF TREATING CANCER USING PYRIDOPYRIMIDINONE INHIBITORS OF PI3K ALPHA
Abstract: The present invention provides methods of treating cancer by administering a compound of Formula I, optionally as a pharmaceutically acceptable salt, solvate and/or hydrate thereof, in combination with other cancer treatments. (Formula I)
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Org. (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (EAPO) (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MT, NL, NO, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (OAPI) (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language:English (EN)
Filing Language:English (EN)

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